SCHEMBL1968189

SCHEMBL1968189

NC(=O)c1cnc(Cl)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 5/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
SIRT6 Q8N6T7 2/20 0.45
LMNA P02545 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MKNK1 Q9BUB5 2/20 0.40
MKNK2 Q9HBH9 2/20 0.40
PARP1 P09874 2/20 0.40
MAP4K4 O95819 2/20 0.40
F7 P08709 1/20 0.40
F3 P13726 1/20 0.40
SARM1 Q6SZW1 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40
SIRT5 Q9NXA8 1/20 0.40
SIRT4 Q9Y6E7 1/20 0.40
NAPRT Q6XQN6 1/20 0.40
JUN P05412 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3407188 0.81 NNMT (0.56) NNMTSMN1; SMN2SIRT6LMNAL3MBTL1
SCHEMBL1745778 0.77 NNMT (0.52) NNMTSMN1; SMN2SIRT6LMNAL3MBTL1
SCHEMBL63857 0.77 NAPRT (0.58) KDM4ENAPRTJUNNFKB1NFKB2
SCHEMBL6987829 0.77 NAPRT (0.46) SMN1; SMN2SIRT6L3MBTL1NAPRTJUN
SCHEMBL3141529 0.77 NNMT (0.58) NNMTSMN1; SMN2SIRT6LMNAL3MBTL1
SCHEMBL669121 0.77 NNMT (0.52) NNMTSMN1; SMN2SIRT6LMNAL3MBTL1
SCHEMBL23193160 0.75 NNMT (0.50) NNMTSMN1; SMN2SIRT6LMNAL3MBTL1
SCHEMBL600134 0.75 NAPRT (0.40) SMN1; SMN2LMNAL3MBTL1KDM4ENAPRT
SCHEMBL388168 0.75 NAPRT (0.67) NNMTSMN1; SMN2SIRT6L3MBTL1KDM4E
SCHEMBL29524193 0.75 NAPRT (0.67) NNMTSMN1; SMN2SIRT6L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110372604-A A kind of synthetic method of the chloro- 5- pyrimidine carboxamide of 2,4- bis- 南京普锐达医药科技有限公司 2019-10-25 CN claimed
WO-2025262297-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 DARK BLUE THERAPEUTICS LTD (GB) 2025-12-26 WO disclosed
EP-4667467-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 Dark Blue Therapeutics Ltd (GB) 2025-12-24 EP disclosed
US-20250326754-A1 DNA-PK Inhibitor Compounds and Uses Thereof ADMARE THERAPEUTICS SOC (CA) 2025-10-23 US disclosed
EP-4522620-A1 DNA-PK INHIBITOR COMPOUNDS AND USES THEREOF Admare Therapeutics Society (CA) 2025-03-19 EP disclosed
US-20240246960-A1 7-Morpholino-L,6-Naphthyridin-5-yl Derivatives and Pharmaceutical Compositions Thereof Useful as DNA-PK Inhibitor PROVINCIAL HEALTH SERVICES AUTHORITY (CA) 2024-07-25 US disclosed
WO-2024054955-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
WO-2024054953-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
WO-2024054954-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
CN-117658992-A Benzimidazole compound, preparation method and pharmaceutical application thereof 中国医学科学院药物研究所 2024-03-08 CN disclosed
CN-104418866-B Dgat1 inhibitor and its preparation method and application 青岛黄海制药有限责任公司 2018-10-16 CN disclosed
WO-2018092089-A1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-05-24 WO disclosed
WO-2018092089-A1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-05-24 WO disclosed
EP-3204363-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE Merck Sharp & Dohme Corp. (US) 2017-08-16 EP disclosed
WO-2016057762-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE MERCK SHARP & DOHME CORP (US) 2016-04-14 WO disclosed
CN-104418866-A DGAT1 inhibitor, and preparation method and application thereof NANJING MINGDE NEW DRUG RES AND DEV CO LTD 2015-03-18 CN disclosed
CN-102348707-A Pyrimidinecarboxamide derivatives as inhibitors of SYK kinase GLAXO GROUP LTD 2012-02-08 CN disclosed
US-20110152295-A1 HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2011-06-23 US disclosed
EP-2334666-A1 HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Canada Inc. (CA) 2011-06-22 EP disclosed
WO-2010025553-A1 HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2010-03-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240246960-A1 7-Morpholino-L,6-Naphthyridin-5-yl Derivatives and Pharmaceutical Compositions Thereof Useful as DNA-PK Inhibitor DCK, ERCC2, POLK NNMT 760/4885SMN1; SMN2 2120/4885SIRT6 1928/4885
US-20250326754-A1 DNA-PK Inhibitor Compounds and Uses Thereof DCK, CHEK1, CHEK2 NNMT 1375/4885SMN1; SMN2 3102/4885SIRT6 1308/4885
US-20110152295-A1 HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE SCD, SCD5, SREBF1 NNMT 810/4885SMN1; SMN2 2669/4885SIRT6 787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.