SCHEMBL3407803

SCHEMBL3407803

COc1cc(Nc2cccc(Nc3ccc(OC(F)(F)F)cc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.43
GALR2 O43603 4/20 0.41
GALR1 P47211 2/20 0.40
ABL1 P00519 7/20 0.39
BCR P11274 6/20 0.39
DHFR P00374 1/20 0.39
BRAF P15056 1/20 0.38
IDH1 O75874 1/20 0.38
CHRNA7 P36544 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408722 0.93 IGF1R (0.52) IGF1RGALR2GALR1BRAFABCB1
SCHEMBL3404287 0.90 GALR2 (0.41) IGF1RGALR2GALR1ABL1BCR
SCHEMBL3404327 0.88 DHODH (0.43) GALR2BRAFABCB1ABCC1ABCG2
SCHEMBL3410817 0.88 GALR2 (0.39) IGF1RGALR2GALR1ABL1BCR
SCHEMBL3406352 0.87 BRAF (0.46) BRAFABCB1ABCC1ABCG2
SCHEMBL3410452 0.87 BRAF (0.44) GALR2GALR1BRAFABCB1ABCC1
SCHEMBL3410067 0.86 IGF1R (0.47) IGF1RGALR2GALR1BRAFABCB1
SCHEMBL3413181 0.85 TP53 (0.48) ABCB1ABCC1ABCG2
SCHEMBL3406368 0.85 BRAF (0.52) ABL1BRAFABCB1ABCC1ABCG2
SCHEMBL3412595 0.82 MAPT (0.41) BRAFABCB1ABCC1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed