SCHEMBL3406352

SCHEMBL3406352

COc1cc(Nc2cccc(Nc3ccc(F)cc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.46
CYP1A2 P05177 3/20 0.46
CYP2D6 P10635 3/20 0.46
CYP2C19 P33261 3/20 0.46
USP2 O75604 2/20 0.46
CYP3A4 P08684 2/20 0.46
TSHR P16473 1/20 0.46
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
PDE4B Q07343 1/20 0.41
PSEN1 P49768 4/20 0.39
PSEN2 P49810 4/20 0.39
APH1B Q8WW43 4/20 0.39
NCSTN Q92542 4/20 0.39
APH1A Q96BI3 4/20 0.39
PSENEN Q9NZ42 4/20 0.39
ABCB1 P08183 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406368 0.94 BRAF (0.52) BRAFCYP1A2CYP2D6CYP2C19USP2
SCHEMBL3410452 0.91 BRAF (0.44) BRAFCYP1A2CYP2D6CYP2C19USP2
SCHEMBL3404327 0.89 DHODH (0.43) BRAFLMNAPSEN1PSEN2APH1B
SCHEMBL3407803 0.87 IGF1R (0.43) BRAFABCB1ABCC1ABCG2
SCHEMBL3412595 0.87 MAPT (0.41) BRAFLMNAPDE4BABCB1ABCC1
SCHEMBL3408722 0.86 IGF1R (0.52) BRAFPSEN1PSEN2APH1BNCSTN
SCHEMBL3413181 0.85 TP53 (0.48) LMNAPSEN1PSEN2APH1BNCSTN
SCHEMBL3413442 0.82 GRM5 (0.41) ABCB1ABCC1ABCG2CDK9CCNT1
SCHEMBL3404331 0.81 ABCB1 (0.41) BRAFPSEN1PSEN2APH1BNCSTN
SCHEMBL3409746 0.81 TP53 (0.47) LMNAPSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed