SCHEMBL3407889

SCHEMBL3407889

Cc1nc(-c2cc3ccccc3o2)c2c(N)c(OC(N)=O)sc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.51
EEF2K O00418 1/20 0.42
PLAU P00749 2/20 0.41
KCNH2 Q12809 1/20 0.41
SCN5A Q14524 1/20 0.41
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
MAPT P10636 6/20 0.37
RAB9A P51151 6/20 0.37
NPC1 O15118 5/20 0.37
SYK P43405 1/20 0.36
F2RL3 Q96RI0 1/20 0.36
TP53 P04637 1/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3411850 0.90 IKBKB (0.48) IKBKBEEF2KPLAUKCNH2SCN5A
SCHEMBL3406686 0.88 IKBKB (0.47) IKBKBEEF2KPLAUKCNH2SCN5A
SCHEMBL1176552 0.84 IKBKB (0.70) IKBKBEEF2KPLAUKCNH2SCN5A
SCHEMBL3414143 0.83 EEF2K (0.42) IKBKBEEF2KMAPTSMN1; SMN2ALDH1A1
SCHEMBL3414021 0.83 IKBKB (0.42) IKBKBEEF2KPLAUKCNH2SCN5A
SCHEMBL3414237 0.81 IKBKB (0.41) IKBKBEEF2KPLAUKCNH2SCN5A
SCHEMBL3412095 0.81 IKBKB (0.47) IKBKBEEF2KPLAUMAPTRAB9A
SCHEMBL3411616 0.80 IKBKB (0.40) IKBKBEEF2KPLAUKCNH2SCN5A
SCHEMBL3657555 0.77 EEF2K (0.46) IKBKBEEF2KPLAUKCNH2SCN5A
SCHEMBL3407940 0.74 EEF2K (0.42) IKBKBEEF2KMAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed