SCHEMBL3414237

SCHEMBL3414237

NC(=O)Oc1sc2nc(-c3cccnc3)nc(-c3cc4ccccc4o3)c2c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.41
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
EEF2K O00418 2/20 0.38
BRAF P15056 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
ALDH1A1 P00352 5/20 0.37
HPGD P15428 3/20 0.37
POLB P06746 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 2/20 0.37
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
RAB9A P51151 2/20 0.36
PLAU P00749 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1176475 0.86 IKBKB (0.56) IKBKBADORA2AADORA1EEF2KBRAF
SCHEMBL3414021 0.84 IKBKB (0.42) IKBKBADORA2AADORA1EEF2KKDM4E
SCHEMBL3411850 0.83 IKBKB (0.48) IKBKBEEF2KBRAFPDE4APDE4B
SCHEMBL3407889 0.81 IKBKB (0.51) IKBKBEEF2KALDH1A1HPGDKDM4E
SCHEMBL3406686 0.80 IKBKB (0.47) IKBKBEEF2KBRAFPDE4APDE4B
SCHEMBL3411616 0.72 IKBKB (0.40) IKBKBEEF2KBRAFPDE4APDE4B
SCHEMBL3657555 0.71 EEF2K (0.46) IKBKBADORA2AEEF2KBRAFALDH1A1
SCHEMBL3413366 0.71 IKBKB (0.41) IKBKBADORA2AADORA1EEF2KALDH1A1
SCHEMBL1176329 0.70 IKBKB (0.58) IKBKBADORA2AADORA1EEF2KBRAF
SCHEMBL12885228 0.70 ALDH1A1 (0.37) ALDH1A1HPGDPOLBKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed