SCHEMBL3407986

SCHEMBL3407986

Cc1ccc(-c2nc(C3CC3)nc3sc(OC(N)=O)c(N)c23)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
MAPT P10636 6/20 0.40
HPGD P15428 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 2/20 0.40
LIMK1 P53667 1/20 0.39
CDK8 P49336 1/20 0.33
CDK19 Q9BWU1 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
ADORA2A P29274 4/20 0.32
ADORA1 P30542 3/20 0.32
GRM1 Q13255 1/20 0.32
ADORA3 P0DMS8 2/20 0.32
ADORA2B P29275 2/20 0.32
KDM4E B2RXH2 3/20 0.31
PKM P14618 1/20 0.31
POLB P06746 1/20 0.31
HSP90AA1 P07900 1/20 0.31
LMNA P02545 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3410981 0.85 LIMK1 (0.42) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL1176092 0.85 HPGD (0.56) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3406840 0.82 LIMK1 (0.42) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3411178 0.82 LHCGR (0.40) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3414147 0.82 LIMK1 (0.42) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3413287 0.81 LIMK1 (0.39) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3410251 0.79 IKBKB (0.41) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3407423 0.76 LIMK1 (0.36) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3409496 0.76 BRAF (0.40) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL3409081 0.76 ADORA2A (0.36) ALDH1A1MAPTHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP claimed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO claimed
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed