SCHEMBL3408742

SCHEMBL3408742

Cc1cccc(-c2nc(N3CCOCC3)nc3sc(OC(N)=O)c(N)c23)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.40
HTT P42858 4/20 0.38
HSD17B10 Q99714 3/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
BRD9 Q9H8M2 1/20 0.37
BAZ2B Q9UIF8 1/20 0.37
HPGD P15428 5/20 0.35
PIK3CA P42336 4/20 0.35
RXFP1 Q9HBX9 2/20 0.35
KDM4E B2RXH2 6/20 0.35
ALDH1A1 P00352 5/20 0.35
MAPT P10636 3/20 0.35
GAA P10253 2/20 0.35
GLA P06280 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1176780 0.86 IKBKB (0.56) IKBKBHTTHSD17B10LMNAPOLB
SCHEMBL3410251 0.83 IKBKB (0.41) IKBKBHTTHSD17B10LMNAPOLB
SCHEMBL3414045 0.81 TGFBR1 (0.37) IKBKBKDM4EALDH1A1MAPTMAPK1
SCHEMBL3407926 0.79 PRKDC (0.43) IKBKBHTTHSD17B10LMNAPOLB
SCHEMBL3411093 0.78 IKBKB (0.34) IKBKBALDH1A1GAATSHRMEN1
SCHEMBL3411826 0.76 IKBKB (0.45) IKBKBLMNAKDM4EALDH1A1GAA
SCHEMBL3410902 0.73 LHCGR (0.35) IKBKB
SCHEMBL3410905 0.73 BRAF (0.33) IKBKBSMN1; SMN2MEN1KMT2A
SCHEMBL3408720 0.71 BRAF (0.35) IKBKB
SCHEMBL3409644 0.71 MEN1 (0.36) HSD17B10HPGDALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP claimed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO claimed
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed