SCHEMBL3409027

SCHEMBL3409027

c1cnc2c(c1)CCCC2NCc1ccc2nc(Cc3nc4ccccc4[nH]3)oc2c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 18/20 0.47
SLC40A1 Q9NP59 1/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
CHRM2 P08172 1/20 0.43
CYP2D6 P10635 1/20 0.43
DRD2 P14416 1/20 0.43
OPRM1 P35372 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408734 0.94 CXCR4 (0.47) CXCR4SLC40A1HDAC1HDAC6CHRM2
SCHEMBL4760828 0.82 SLC40A1 (0.59) CXCR4SLC40A1CHRM2CYP2D6DRD2
SCHEMBL31257251 0.82 SLC40A1 (0.59) CXCR4SLC40A1CHRM2CYP2D6DRD2
SCHEMBL3370850 0.82 SLC40A1 (0.59) CXCR4SLC40A1CHRM2CYP2D6DRD2
SCHEMBL31059309 0.82 CXCR4 (0.61) CXCR4
SCHEMBL7104696 0.82 CXCR4 (0.61) CXCR4
SCHEMBL3406461 0.79 CXCR4 (0.56) CXCR4SLC40A1CHRM2CYP2D6DRD2
SCHEMBL4069397 0.77 CXCR4 (0.76) CXCR4CHRM2CYP2D6DRD2OPRM1
Bromide SCHEMBL5140662 0.76 CXCR4 (0.75) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL7074716 0.75 SLC40A1 (0.63) CXCR4SLC40A1CHRM2CYP2D6DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1752455-B1 Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2010-11-10 EP claimed