SCHEMBL3409713

SCHEMBL3409713

COc1cc(Nc2nc(C3CC3)cc(C(C)(C)O)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.36
EHMT2 Q96KQ7 2/20 0.35
EHMT1 Q9H9B1 1/20 0.35
PSEN1 P49768 2/20 0.34
PSEN2 P49810 2/20 0.34
APH1B Q8WW43 2/20 0.34
NCSTN Q92542 2/20 0.34
APH1A Q96BI3 2/20 0.34
PSENEN Q9NZ42 2/20 0.34
IMPDH2 P12268 6/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PDE7A Q13946 2/20 0.34
ULK1 O75385 1/20 0.33
ULK2 Q8IYT8 1/20 0.33
KCNH2 Q12809 1/20 0.33
CYP17A1 P05093 1/20 0.32
IMPDH1 P20839 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408862 0.87 NPC1 (0.43) EHMT2EHMT1IMPDH2NPC1RAB9A
SCHEMBL3410560 0.86 NPC1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3410112 0.84 PSEN1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3411934 0.83 CDK1 (0.35) EHMT2EHMT1PSEN1PSEN2APH1B
SCHEMBL3411116 0.83 KCNH2 (0.49) EHMT2EHMT1IMPDH2NPC1RAB9A
SCHEMBL3408737 0.83 RET (0.41) ULK1ULK2
SCHEMBL3410528 0.83 GALR2 (0.42)
SCHEMBL3412580 0.82 GALR2 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3409722 0.82 PIK3CA (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3409733 0.82 CDK9 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed