SCHEMBL3409722

SCHEMBL3409722

COc1cc(Nc2nc(-c3ccc(Cl)cc3)cc(C(C)(C)O)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.41
PIK3CB P42338 2/20 0.41
PIK3CG P48736 2/20 0.41
JAK2 O60674 1/20 0.41
EGFR P00533 1/20 0.41
CDK2 P24941 1/20 0.41
PTK2B Q14289 1/20 0.41
PSEN1 P49768 2/20 0.41
PSEN2 P49810 2/20 0.41
APH1B Q8WW43 2/20 0.41
NCSTN Q92542 2/20 0.41
APH1A Q96BI3 2/20 0.41
PSENEN Q9NZ42 2/20 0.41
AGPAT2 O15120 4/20 0.40
ALOX5 P09917 1/20 0.40
CXCL12 P48061 1/20 0.38
MAPT P10636 6/20 0.38
IMPDH2 P12268 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3412384 0.90 AGPAT2 (0.41) PIK3CAPIK3CBPIK3CGPSEN1PSEN2
SCHEMBL3407100 0.90 MAPT (0.48) PIK3CAPIK3CBPIK3CGJAK2EGFR
SCHEMBL3412354 0.90 PTGS2 (0.39) JAK2PSEN1PSEN2APH1BNCSTN
SCHEMBL3406823 0.87 NPC1 (0.39) AGPAT2MAPTIMPDH2SMN1; SMN2NPC1
SCHEMBL3405215 0.87 KCNH2 (0.37) CDK2IMPDH2NPC1RAB9APTGS2
SCHEMBL3413207 0.87 PSEN1 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3408862 0.86 NPC1 (0.43) IMPDH2NPC1RAB9A
SCHEMBL3410560 0.85 NPC1 (0.37) CDK2PSEN1PSEN2APH1BNCSTN
SCHEMBL3407305 0.83 PIK3CA (0.61) PIK3CAPIK3CBPIK3CGJAK2EGFR
SCHEMBL3406534 0.83 SYK (0.39) JAK2IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed