SCHEMBL3413176

SCHEMBL3413176

O=C(Nc1ccc2nc(N[C@@H]3CCc4ccccc43)ccc2c1)N(C1CCCCC1)N(C(=O)Nc1ccc2nc(N[C@@H]3CCc4ccccc43)ccc2c1)C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
HPGDS O60760 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
JAK3 P52333 1/20 0.37
PFKFB3 Q16875 3/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FADS1 O60427 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
MCHR1 Q99705 1/20 0.36
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3409104 0.84 HPGDS (0.39) NPC1RAB9AALDH1A1HTTHPGDS
SCHEMBL3404457 0.84 RAB9A (0.47) NPC1RAB9AHPGDSJAK2JAK1
SCHEMBL3413540 0.84 RAB9A (0.50) NPC1RAB9AALDH1A1JAK2JAK1
SCHEMBL4109902 0.83 MAPT (0.44) NPC1RAB9AALDH1A1HPGDSJAK2
SCHEMBL3414984 0.83 AURKA (0.41) NPC1HPGDSJAK2JAK1TYK2
SCHEMBL3403165 0.82 KMT2A (0.48) NPC1RAB9AALDH1A1HPGDSLMNA
SCHEMBL3415639 0.82 NPC1 (0.47) NPC1RAB9AKDM4ETSHRSMN1; SMN2
SCHEMBL3398520 0.82 RAB9A (0.38) NPC1RAB9AALDH1A1HTTHPGDS
SCHEMBL3415257 0.82 HPGDS (0.46) NPC1RAB9AALDH1A1HPGDSJAK2
SCHEMBL3411790 0.82 NPC1 (0.42) NPC1ALDH1A1HPGDSJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262789-A1 2-AMINOQUINOLINES F. Hoffmann-La Roche AG (CH) 2010-12-22 EP disclosed
WO-2009109477-A1 2-AMINOQUINOLINES F. HOFFMANN-LA ROCHE AG (CH) 2009-09-11 WO disclosed