SCHEMBL3413379

SCHEMBL3413379

CC(C)(C)c1nc(-c2ccco2)c2c(N)c(OC(N)=O)sc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.43
LIMK1 P53667 1/20 0.41
MAPT P10636 8/20 0.38
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 4/20 0.38
HPGD P15428 3/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
RECQL P46063 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MCL1 Q07820 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
LMNA P02545 1/20 0.38
HSD17B10 Q99714 5/20 0.38
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
HTT P42858 2/20 0.38
THRB P10828 2/20 0.38
GFER P55789 1/20 0.38
ESR2 Q92731 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3412095 0.86 IKBKB (0.47) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL3407525 0.86 LIMK1 (0.45) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL3408796 0.84 IKBKB (0.43) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL1176582 0.84 IKBKB (0.61) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL3406906 0.83 MAPT (0.45) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL3414147 0.83 LIMK1 (0.42) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL3408735 0.82 IKBKB (0.42) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL3411093 0.81 IKBKB (0.34) IKBKBLIMK1ALDH1A1MEN1KMT2A
SCHEMBL3409501 0.77 IKBKB (0.44) IKBKBLIMK1MAPTKDM4EALDH1A1
SCHEMBL5732361 0.74 LIMK1 (0.50) IKBKBLIMK1MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed