SCHEMBL3407525

SCHEMBL3407525

NC(=O)Oc1sc2nc(N)nc(-c3ccco3)c2c1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 1/20 0.45
IKBKB O14920 1/20 0.44
MAPT P10636 7/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 4/20 0.41
HPGD P15428 3/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RECQL P46063 2/20 0.41
MCL1 Q07820 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
LMNA P02545 1/20 0.41
ADORA2A P29274 7/20 0.41
ADORA1 P30542 6/20 0.41
HSD17B10 Q99714 4/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
HTT P42858 2/20 0.41
USP2 O75604 1/20 0.41
PTK2B Q14289 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3412095 0.89 IKBKB (0.47) LIMK1IKBKBMAPTALDH1A1KDM4E
SCHEMBL3408796 0.87 IKBKB (0.43) LIMK1IKBKBMAPTALDH1A1KDM4E
SCHEMBL3413379 0.86 IKBKB (0.43) LIMK1IKBKBMAPTALDH1A1KDM4E
SCHEMBL3406906 0.86 MAPT (0.45) LIMK1IKBKBMAPTALDH1A1KDM4E
SCHEMBL3408735 0.85 IKBKB (0.42) LIMK1IKBKBMAPTALDH1A1KDM4E
SCHEMBL1175798 0.82 IKBKB (0.64) LIMK1IKBKBMAPTALDH1A1KDM4E
SCHEMBL3410981 0.81 LIMK1 (0.42) LIMK1MAPTALDH1A1KDM4EHPGD
SCHEMBL3411850 0.80 IKBKB (0.48) LIMK1IKBKBMAPTNPC1RAB9A
SCHEMBL3409501 0.80 IKBKB (0.44) LIMK1IKBKBMAPTALDH1A1KDM4E
SCHEMBL3414045 0.78 TGFBR1 (0.37) LIMK1IKBKBMAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP claimed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO claimed
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed