SCHEMBL3409501

SCHEMBL3409501

Cc1cc(C)n(-c2nc(-c3ccco3)c3c(N)c(OC(N)=O)sc3n2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.44
KDM4E B2RXH2 6/20 0.39
MAPT P10636 5/20 0.39
HSD17B10 Q99714 5/20 0.39
ALDH1A1 P00352 5/20 0.39
HPGD P15428 4/20 0.39
POLB P06746 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALOX15 P16050 2/20 0.39
BLM P54132 2/20 0.39
PKM P14618 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LIMK1 P53667 1/20 0.39
ADORA2A P29274 3/20 0.36
ADORA1 P30542 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1176569 0.86 IKBKB (0.61) IKBKBKDM4EMAPTHSD17B10ALDH1A1
SCHEMBL3411618 0.85 EEF2K (0.39) KDM4EMAPTHSD17B10ALDH1A1HPGD
SCHEMBL3412095 0.82 IKBKB (0.47) IKBKBKDM4EMAPTHSD17B10ALDH1A1
SCHEMBL3407525 0.80 LIMK1 (0.45) IKBKBKDM4EMAPTHSD17B10ALDH1A1
SCHEMBL3408796 0.78 IKBKB (0.43) IKBKBKDM4EMAPTHSD17B10ALDH1A1
SCHEMBL3406906 0.77 MAPT (0.45) IKBKBKDM4EMAPTHSD17B10ALDH1A1
SCHEMBL3413379 0.77 IKBKB (0.43) IKBKBKDM4EMAPTHSD17B10ALDH1A1
SCHEMBL3408735 0.76 IKBKB (0.42) IKBKBKDM4EMAPTHSD17B10ALDH1A1
SCHEMBL1176022 0.70 EEF2K (0.53) IKBKBKDM4EMAPTALDH1A1HPGD
SCHEMBL3408742 0.70 IKBKB (0.40) IKBKBKDM4EMAPTHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP claimed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO claimed
EP-2260044-A2 THIENOPYRIMIDINES Merck Patent GmbH (DE) 2010-12-15 EP disclosed
WO-2009124653-A2 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2009-10-15 WO disclosed