SCHEMBL3418495

SCHEMBL3418495

COCCCOc1cc(CN(C(=O)[C@H]2CNCC[C@]2(O)c2ccc(F)c(F)c2)C2CC2)c(Cl)cn1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
REN P00797 20/20 0.75
KCNH2 Q12809 15/20 0.75
CYP3A4 P08684 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3112098 0.90 REN (0.78) RENKCNH2CYP3A4
SCHEMBL3112119 0.90 REN (0.78) RENKCNH2CYP3A4
SCHEMBL3108094 0.85 REN (1.00) RENKCNH2CYP3A4
SCHEMBL3108124 0.85 REN (1.00) RENKCNH2CYP3A4
SCHEMBL3105676 0.85 REN (1.00) RENKCNH2CYP3A4
SCHEMBL3105660 0.85 REN (1.00) RENKCNH2CYP3A4
SCHEMBL3418490 0.84 REN (0.70) RENKCNH2CYP3A4
SCHEMBL3097101 0.82 REN (0.65) RENKCNH2CYP3A4
SCHEMBL3107698 0.82 REN (0.76) RENKCNH2CYP3A4
SCHEMBL3109779 0.82 REN (0.76) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229363-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2010-09-22 EP claimed
WO-2009070869-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-06-11 WO claimed
EP-2229363-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2010-09-22 EP disclosed
WO-2009070869-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-06-11 WO disclosed