Benzoclidine

Benzoclidine

SCHEMBL342347

O=C(OC1CN2CCC1CC2)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.74
TSHR P16473 1/20 0.69
RXFP1 Q9HBX9 1/20 0.69
CYP2D6 P10635 1/20 0.68
CHRNA7 P36544 3/20 0.65
BCHE P06276 1/20 0.65
ACHE P22303 1/20 0.65
MEN1 O00255 1/20 0.64
KMT2A Q03164 1/20 0.64
CHRM3 P20309 6/20 0.63
CHRM2 P08172 5/20 0.63
CHRM1 P11229 5/20 0.63
CHRM4 P08173 1/20 0.62
CHRM5 P08912 1/20 0.62
HTR3E A5X5Y0 1/20 0.60
HTR3B O95264 1/20 0.60
CHRNB2 P17787 1/20 0.60
CHRNA4 P43681 1/20 0.60
HTR3A P46098 1/20 0.60
HTR3D Q70Z44 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzoclidine SCHEMBL1542330 1.00 GLA (0.74) GLATSHRRXFP1CYP2D6CHRNA7
Benzoclidine SCHEMBL1542430 1.00 GLA (0.74) GLATSHRRXFP1CYP2D6CHRNA7
SCHEMBL1234895 0.85 CYP2D6 (0.65) TSHRRXFP1CYP2D6CHRNA7BCHE
SCHEMBL1234896 0.85 CYP2D6 (0.65) TSHRRXFP1CYP2D6CHRNA7BCHE
Bicarbonate SCHEMBL1721399 0.83 GLA (0.67) GLATSHRRXFP1CYP2D6CHRNA7
Bicarbonate SCHEMBL1720584 0.83 GLA (0.67) GLATSHRRXFP1CYP2D6CHRNA7
SCHEMBL7824053 0.82 CYP2D6 (0.62) TSHRRXFP1CYP2D6CHRNA7BCHE
SCHEMBL7824049 0.82 CYP2D6 (0.62) TSHRRXFP1CYP2D6CHRNA7BCHE
SCHEMBL11896515 0.82 GLA (0.58) GLATSHRRXFP1CYP2D6CHRNA7
SCHEMBL8935124 0.81 CHRNA7 (0.60) GLATSHRRXFP1CHRNA7BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 129 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118638109-A Preparation method of opium drug-oxelidine 中山大学 2024-09-13 CN claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-1605939-B1 PHARMACEUTICAL USE OF 1-AZABICYCLO¬ 2.2.2 OCTANES AND A METHOD OF TESTING COMPOUNDS FOR THE ABILITY OF ACTIVATING INACTIVE WT P53 APREA AB (SE) 2008-10-15 EP claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20060276502-A1 Pharmaceutical use of 1-azabicyclo[2.2.2]octanes and a method of testing compounds for the ability of activating inactive wt p53. APREA AB (SE) 2006-12-07 US claimed
EP-1476166-B1 USE OF LOW MOLECULAR WEIGHT COMPOUNDS FOR PREPARING A MEDICAMENT USEFUL IN TREATING MUTANT P53 MEDIATED DISEASES APREA AB (SE) 2006-07-19 EP claimed
EP-1605939-A1 PHARMACEUTICAL USE OF 1-AZABICYCLO[ 2.2.2] OCTANES AND A METHOD OF TESTING COMPOUNDS FOR THE ABILITY OF ACTIVATING INACTIVE WT P53 APREA AB (SE) 2005-12-21 EP claimed
US-20050090510-A1 Use of low molecular weight compounds for preparing a medicament useful in treating mutant p53 mediated diseases APREA THERAPEUTICS AB (SE) 2005-04-28 US claimed
EP-1476166-A1 USE OF LOW MOLECULAR WEIGHT COMPOUNDS FOR PREPARING A MEDICAMENT USEFUL IN TREATING MUTANT P53 MEDIATED DISEASES APREA AB (SE) 2004-11-17 EP claimed
WO-2004084893-A1 PHARMACEUTICAL USE OF 1-AZABICYCLO[2.2.2]OCTANES AND A METHOD OF TESTING COMPOUNDS FOR THE ABILITY OF ACTIVATING INACTIVE WT P53 APREA AB (SE) 2004-10-07 WO claimed
WO-2003070250-A1 USE OF LOW MOLECULAR WEIGHT COMPOUNDS FOR PREPARING A MEDICAMENT USEFUL IN TREATING MUTANT P53 MEDIATED DISEASES APREA AB (SE) 2003-08-28 WO claimed
US-4835162-A 3-QUINUCLIDINYL BENZOATE OR METHYL CARBAMATE UNIVERSITY OF ROCHESTER 1989-05-30 US claimed
CN-118638109-B Preparation method of opium drug-oxelidine 中山大学 2025-10-28 CN disclosed
CN-118638109-B Preparation method of opium drug-oxelidine 中山大学 2025-10-28 CN disclosed
US-4966916-A DI-AND TRIMETHYLAMINOETHYL BENZOATES, PHENYLCARBAMATES AND PHENYLTHIOCARBAMATES UNIVERSITY OF ROCHESTER 1990-10-30 US disclosed
EP-0347844-A2 A translucent cosmetic emulsion KAO CORPORATION (JP) 1989-12-27 EP disclosed
US-4835162-A 3-QUINUCLIDINYL BENZOATE OR METHYL CARBAMATE UNIVERSITY OF ROCHESTER 1989-05-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276502-A1 Pharmaceutical use of 1-azabicyclo[2.2.2]octanes and a method of testing compounds for the ability of activating inactive wt p53. TP53, TP53BP1, MITF GLA 438/4885TSHR 1582/4885RXFP1 3490/4885
US-20050090510-A1 Use of low molecular weight compounds for preparing a medicament useful in treating mutant p53 mediated diseases TP53, ACP1, TP53BP1 GLA 1144/4885TSHR 3751/4885RXFP1 4528/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.