SCHEMBL3424926

SCHEMBL3424926

Cc1cccc(-n2ncc3c(Cl)ncnc32)c1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 11/20 0.54
FSCN1 Q16658 1/20 0.50
MAPT P10636 5/20 0.47
SLC2A1 P11166 1/20 0.44
SLC2A2 P11168 1/20 0.44
SLC2A3 P11169 1/20 0.44
RAB9A P51151 3/20 0.43
LMNA P02545 6/20 0.43
GSK3B P49841 1/20 0.42
NPC1 O15118 2/20 0.42
HTT P42858 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPBWR1 P48145 1/20 0.42
MCHR1 Q99705 1/20 0.42
PDE9A O76083 1/20 0.42
KDM4E B2RXH2 1/20 0.41
BLM P54132 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL839442 0.89 TP53 (0.46) TP53FSCN1MAPTSLC2A1SLC2A2
SCHEMBL839657 0.89 SLC2A1 (0.54) TP53FSCN1MAPTSLC2A1SLC2A2
SCHEMBL838678 0.86 TP53 (0.44) TP53FSCN1MAPTSLC2A1SLC2A2
SCHEMBL839711 0.83 SLC2A1 (0.47) TP53FSCN1MAPTSLC2A1SLC2A2
SCHEMBL838336 0.81 TP53 (0.41) TP53MAPTSLC2A1SLC2A2SLC2A3
SCHEMBL838829 0.80 P2RX7 (0.46) TP53MAPTRAB9ALMNANPC1
SCHEMBL839210 0.80 GCK (0.47) TP53MAPTSLC2A1SLC2A2SLC2A3
SCHEMBL838694 0.78 CYP17A1 (0.46) TP53MAPTRAB9ALMNAGSK3B
SCHEMBL839601 0.78 RAB9A (0.55) TP53MAPTRAB9ALMNANPC1
SCHEMBL838498 0.78 RAB9A (0.46) TP53MAPTRAB9ALMNAGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247596-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS Natco Pharma Limited (IN) 2010-11-10 EP disclosed
WO-2009098715-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS NATCO PHARMA LIMITED (IN) 2009-08-13 WO disclosed