SCHEMBL3425640

SCHEMBL3425640

Cc1ccc(C2=CN=CCN2C#N)cc1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 2/20 0.33
MAPT P10636 2/20 0.33
RAB9A P51151 2/20 0.33
GFER P55789 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ERBB2 P04626 1/20 0.33
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
CYP2A6 P11509 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PTAFR P25105 1/20 0.30
NTRK1 P04629 1/20 0.30
PIM1 P11309 1/20 0.30
ACVR1 Q04771 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9137525 0.67
SCHEMBL13258567 0.61 NISCH (0.36) KMT2ANPC1MAPTRAB9AGFER
SCHEMBL21697025 0.61 PDE3B (0.33) KMT2ANPC1MAPTRAB9ASMN1; SMN2
Water SCHEMBL3680095 0.58 ACHE (0.67) ALDH1A1HPGDCYP2A6HSD17B10
Water SCHEMBL3763584 0.58 ACHE (0.67) ALDH1A1HPGDCYP2A6HSD17B10
P-Xylene SCHEMBL1443687 0.56 ACHE (0.61) KMT2ANPC1MAPTRAB9AALDH1A1
SCHEMBL197731 0.55 ACHE (0.73) ALDH1A1HPGDHSD17B10
SCHEMBL18661495 0.55 ACHE (0.73) ALDH1A1HPGDHSD17B10
SCHEMBL3287696 0.55 ACHE (0.73) ALDH1A1HPGDHSD17B10
P-Xylene SCHEMBL18229935 0.55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247586-A1 2-AZA-BICYCLO[2.2.1]HEPTANE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2010-11-10 EP disclosed
WO-2009104155-A1 2-AZA-BICYCLO[2.2.1]HEPTANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2009-08-27 WO disclosed