SCHEMBL3428537

SCHEMBL3428537

N#Cc1cc(C(Cl)(Cl)Cl)cnc1Cl

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
NPSR1 Q6W5P4 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
KHK P50053 1/20 0.37
KDM4E B2RXH2 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP11B2 P19099 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2634852 0.83 ALDH1A1 (0.49) ALDH1A1NPSR1TDP1KHKKDM4E
SCHEMBL21338969 0.83 ALDH1A1 (0.49) ALDH1A1NPSR1TDP1KHKKDM4E
SCHEMBL30055347 0.83 ALDH1A1 (0.49) ALDH1A1NPSR1TDP1KHKKDM4E
SCHEMBL1031743 0.75 ALDH1A1 (0.56) ALDH1A1NPSR1TDP1KHKKDM4E
SCHEMBL30681117 0.75 ALDH1A1 (0.56) ALDH1A1NPSR1TDP1KHKKDM4E
SCHEMBL7216099 0.74 ALDH1A1 (0.55) ALDH1A1NPSR1TDP1KHKKDM4E
SCHEMBL30681150 0.74 ALDH1A1 (0.55) ALDH1A1NPSR1TDP1KHKKDM4E
SCHEMBL1747710 0.73 TSHR (0.44) ALDH1A1NPSR1TDP1KDM4ESMN1; SMN2
SCHEMBL29504068 0.73 TSHR (0.44) ALDH1A1NPSR1TDP1KDM4ESMN1; SMN2
SCHEMBL1164261 0.72 ALDH1A1 (0.53) ALDH1A1NPSR1TDP1KHKCSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759459-B2 Fluorescent assays for protein kinases ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2010-07-20 US disclosed
US-20050054024-A1 Fluorescent assays for protein kinases NATIONAL INSTITUTES OF HEALTH 2005-03-10 US disclosed
WO-2004062475-A2 FLUORESCENT ASSAYS FOR PROTEIN KINASES ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2004-07-29 WO disclosed