SCHEMBL3429460

SCHEMBL3429460

CCOC(=O)Oc1cc(-c2cc(F)cc(OC)c2)n(-c2ccc(F)c(Cl)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPA1 P27694 1/20 0.41
SLC16A3 O15427 4/20 0.40
SLC16A1 P53985 4/20 0.40
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
KDR P35968 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
POLB P06746 2/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
ALDH1A1 P00352 2/20 0.38
ALOX5 P09917 1/20 0.37
PTGS2 P35354 1/20 0.37
BRD9 Q9H8M2 1/20 0.37
MDM2 Q00987 1/20 0.36
MALT1 Q9UDY8 1/20 0.36
MARS1 P56192 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3427741 0.91 RXFP1 (0.41) RPA1RXRARXRBRXRGKDR
SCHEMBL3428152 0.90 SLC16A3 (0.50) SLC16A3SLC16A1RXRARXRBRXRG
SCHEMBL3429822 0.88 RXFP1 (0.39) RPA1RXRARXRBRXRGKDR
SCHEMBL3427568 0.88 RPA1 (0.46) RPA1SLC16A3SLC16A1RXRARXRB
SCHEMBL3430605 0.86 RXFP1 (0.43) RPA1RXFP1POLBALDH1A1BRD9
SCHEMBL3427610 0.86 RPA1 (0.45) RPA1KDRRXFP1POLBALDH1A1
SCHEMBL3434352 0.86 RPA1 (0.39) RPA1RXRARXRBRXRGKDR
SCHEMBL1764893 0.85 CHRNA7 (0.51) RPA1RXFP1POLBTP53MALT1
SCHEMBL3431941 0.82 ALDH1A1 (0.45) SLC16A3SLC16A1RXRARXRBRXRG
SCHEMBL3423931 0.81 SLC5A1 (0.47) RPA1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed