SCHEMBL3429697

SCHEMBL3429697

CNS(=O)(=O)CCNC(=O)c1cccc(-c2cccc(Oc3cc(Cl)cc(Cl)c3)n2)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 2/20 0.48
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MCL1 Q07820 3/20 0.41
BCL2L1 Q07817 2/20 0.41
LOX P28300 2/20 0.39
LOXL2 Q9Y4K0 2/20 0.39
GRM5 P41594 2/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
SCN9A Q15858 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL958467 0.85 GPR52 (0.63) GPR52MCL1BCL2L1GRM5
SCHEMBL957800 0.83 GPR52 (0.50) GPR52NPC1RAB9AMCL1BCL2L1
SCHEMBL958528 0.83 GPR52 (0.56) GPR52MCL1BCL2L1LOXL2GRM5
SCHEMBL957908 0.82 GPR52 (0.49) GPR52MCL1BCL2L1GRM5NR1H2
SCHEMBL964557 0.82 GPR52 (0.50) GPR52MCL1BCL2L1LOXL2GRM5
SCHEMBL961526 0.79 MAP4K4 (0.56) GPR52
SCHEMBL964554 0.78 LOX (0.49) GPR52MCL1BCL2L1LOXLOXL2
SCHEMBL958267 0.77 L3MBTL1 (0.60) GPR52NPC1RAB9AGRM5NR1H2
SCHEMBL961657 0.77 MAP4K4 (0.53) GPR52NPC1RAB9AMCL1BCL2L1
SCHEMBL959832 0.76 GPR52 (0.46) GPR52MCL1BCL2L1GRM5SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253618-A1 COMPOUND HAVING 6-MEMBERED AROMATIC RING Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed