SCHEMBL3429941

SCHEMBL3429941

C[Si](C)(C)C#Cc1cccc(-n2cccn2)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
NOTUM Q6P988 1/20 0.40
GRM5 P41594 4/20 0.40
ERCC1 P07992 1/20 0.39
ERCC4 Q92889 1/20 0.39
KAT6A Q92794 2/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPK1 P28482 2/20 0.37
HCRTR1 O43613 3/20 0.35
HCRTR2 O43614 3/20 0.35
MPO P05164 1/20 0.34
MAPT P10636 3/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
G6PD P11413 1/20 0.34
KMT2A Q03164 1/20 0.34
NPC1 O15118 1/20 0.34
PDK2 Q15119 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25614598 0.81 KDM4E (0.40) LMNANOTUMGRM5KDM4EALDH1A1
SCHEMBL31635838 0.78 LMNA (0.40) LMNANOTUMGRM5ERCC1ERCC4
SCHEMBL4702337 0.78 GRM5 (0.55) LMNANOTUMGRM5KDM4EALDH1A1
SCHEMBL27822298 0.78 NOTUM (0.44) LMNANOTUMGRM5ERCC1ERCC4
SCHEMBL31635842 0.77 LMNA (0.38) LMNANOTUMGRM5ERCC1ERCC4
SCHEMBL5934873 0.76 NOTUM (0.57) LMNANOTUMGRM5ERCC1ERCC4
SCHEMBL31635836 0.74 KAT6A (0.38) LMNANOTUMGRM5ERCC1ERCC4
Hydrochloric Acid SCHEMBL6006151 0.74 NOTUM (0.55) LMNANOTUMGRM5ERCC1ERCC4
SCHEMBL3614755 0.74 GRM5 (0.39) GRM5KDM4EALDH1A1MEN1KMT2A
SCHEMBL18946125 0.72 DRD2 (0.44) GRM5KDM4EALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247596-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS Natco Pharma Limited (IN) 2010-11-10 EP claimed
WO-2009098715-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS NATCO PHARMA LIMITED (IN) 2009-08-13 WO claimed