SCHEMBL3430002

SCHEMBL3430002

O=C(Nc1ccncc1)N(c1ccccc1)c1cncnc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
JAK2 O60674 2/20 0.49
TYK2 P29597 2/20 0.49
HTT P42858 3/20 0.45
MDM2 Q00987 1/20 0.44
POLB P06746 2/20 0.44
STAT3 P40763 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
BCAT2 O15382 1/20 0.44
LMNA P02545 3/20 0.43
ALDH1A1 P00352 2/20 0.42
HSD17B10 Q99714 1/20 0.42
EPHX1 P07099 1/20 0.42
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3426753 0.94 MEN1 (0.54) TAAR1MEN1KMT2AHTTSMN1; SMN2
SCHEMBL10536719 0.91 TAAR1 (0.61) TAAR1MEN1KMT2AJAK2TYK2
SCHEMBL3429719 0.86 HTT (0.47) MEN1KMT2AHTTROCK2ROCK1
SCHEMBL3429605 0.85 NPC1 (0.56) MEN1KMT2ASMN1; SMN2LMNAALDH1A1
SCHEMBL3430925 0.83 MEN1 (0.44) MEN1KMT2AHTTSMN1; SMN2BCAT2
SCHEMBL3427447 0.83 GRM5 (0.49) MEN1KMT2ASMN1; SMN2
SCHEMBL3428051 0.83 MEN1 (0.50) MEN1KMT2APOLBSMN1; SMN2ALDH1A1
SCHEMBL2533213 0.82 MEN1 (0.49) TAAR1MEN1KMT2AJAK2TYK2
SCHEMBL3430947 0.80 NPC1 (0.44) MEN1KMT2AHTTSMN1; SMN2BCAT2
SCHEMBL1382899 0.80 MEN1 (0.67) TAAR1MEN1KMT2AHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252296-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES Wyeth LLC (US) 2010-11-24 EP disclosed
WO-2009091788-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-07-23 WO disclosed