SCHEMBL3428051

SCHEMBL3428051

O=C(Nc1ccc([N+](=O)[O-])cc1)N(c1ccccc1)c1cncnc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.50
KMT2A Q03164 6/20 0.50
POLB P06746 3/20 0.50
MITF O75030 2/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
GAA P10253 1/20 0.50
HSP90AA1 P07900 1/20 0.47
PTGES O14684 1/20 0.46
CYP19A1 P11511 1/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NAMPT P43490 1/20 0.46
MAPT P10636 3/20 0.45
MAPK1 P28482 2/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MYOC Q99972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3426753 0.85 MEN1 (0.54) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL3430002 0.83 TAAR1 (0.51) MEN1KMT2APOLBALDH1A1SMN1; SMN2
SCHEMBL3429605 0.78 NPC1 (0.56) MEN1KMT2ANPC1RAB9AGAA
SCHEMBL3429719 0.76 HTT (0.47) MEN1KMT2ANAMPT
SCHEMBL3430925 0.75 MEN1 (0.44) MEN1KMT2ANPC1RAB9AGAA
SCHEMBL8325952 0.75 CYP19A1 (0.46) MEN1KMT2ANPC1RAB9ACYP19A1
SCHEMBL3431685 0.74 LTA4H (0.56) MEN1KMT2AALDH1A1NAMPTMAPT
SCHEMBL3434704 0.73 NPC1 (0.55) MEN1KMT2ANPC1RAB9AGAA
SCHEMBL10536719 0.73 TAAR1 (0.61) MEN1KMT2APOLBALDH1A1SMN1; SMN2
SCHEMBL11853543 0.73 MEN1 (0.60) MEN1KMT2APOLBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252296-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES Wyeth LLC (US) 2010-11-24 EP disclosed
WO-2009091788-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-07-23 WO disclosed