SCHEMBL3430947

SCHEMBL3430947

O=C(Nc1cccs1)N(c1ccccc1)c1cncnc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.44
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
GBA1 P04062 1/20 0.39
GAA P10253 11/20 0.39
MEN1 O00255 9/20 0.39
KMT2A Q03164 9/20 0.39
MAPT P10636 7/20 0.39
HSD17B10 Q99714 6/20 0.39
HTT P42858 5/20 0.39
ALOX15 P16050 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPK1 P28482 2/20 0.39
TP53 P04637 2/20 0.39
HPGD P15428 2/20 0.39
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3430002 0.80 TAAR1 (0.51) CA1CA2MEN1KMT2AHSD17B10
SCHEMBL3434055 0.80 RAB9A (0.52) NPC1CA1CA2GAAMEN1
SCHEMBL3426753 0.80 MEN1 (0.54) NPC1CA1CA2MEN1KMT2A
SCHEMBL3430925 0.78 MEN1 (0.44) NPC1CA1CA2GAAMEN1
SCHEMBL3429605 0.75 NPC1 (0.56) NPC1GAAMEN1KMT2AHSD17B10
SCHEMBL6688096 0.74 HPGD (0.49) NPC1GAAMEN1KMT2ASMN1; SMN2
SCHEMBL18825696 0.72 NAMPT (0.50) NPC1GBA1GAAMEN1KMT2A
SCHEMBL7658804 0.71 GAA (0.43) NPC1GBA1GAAMEN1KMT2A
SCHEMBL7658797 0.71 KDM4E (0.46) NPC1GBA1GAAMEN1KMT2A
SCHEMBL9547581 0.71 GAA (0.51) NPC1GAAMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252296-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES Wyeth LLC (US) 2010-11-24 EP disclosed
WO-2009091788-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-07-23 WO disclosed