Apigenin

Apigenin

SCHEMBL3430874

O=c1cc(-c2ccc(O)cc2)oc2cc(O)cc(O)c12.O=c1cc(-c2ccccc2)oc2ccccc12

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.78
MAPT P10636 8/20 0.78
SMN1; SMN2 Q16637 7/20 0.78
ABCB1 P08183 7/20 0.78
CYP1B1 Q16678 7/20 0.78
MEN1 O00255 7/20 0.78
KMT2A Q03164 7/20 0.78
FTO Q9C0B1 6/20 0.78
CYP1A2 P05177 6/20 0.78
CYP19A1 P11511 5/20 0.78
HPGD P15428 5/20 0.78
ABCG2 Q9UNQ0 5/20 0.78
MAOA P21397 5/20 0.78
MAOB P27338 5/20 0.78
TP53 P04637 5/20 0.78
ALDH1A1 P00352 5/20 0.78
CYP1A1 P04798 5/20 0.78
CYP2C9 P11712 5/20 0.78
CYP2C19 P33261 5/20 0.78
KDM4E B2RXH2 4/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chrysin SCHEMBL3858957 0.96 ABCB1 (0.84) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Apigenin SCHEMBL3860131 0.92 CYP3A4 (0.91) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Luteolin SCHEMBL30913900 0.92 POLH (0.75) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Luteolin SCHEMBL15271260 0.92 POLH (0.75) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Luteolin SCHEMBL1229732 0.92 POLH (0.75) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Chrysin SCHEMBL5461671 0.90 CYP3A4 (0.82) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Acacetin SCHEMBL2146352 0.89 MAPT (0.79) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Genkwanin SCHEMBL2464219 0.89 CYP3A4 (0.80) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Chrysin SCHEMBL29383577 0.88 MAPT (1.00) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1
Chrysin SCHEMBL44474 0.88 MAPT (1.00) CYP3A4MAPTSMN1; SMN2ABCB1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4156973-A1 NUTRACEUTICAL COMPOSITION METACEUTIC APS (DK) 2023-04-05 EP claimed
WO-2021239614-A1 NUTRACEUTICAL COMPOSITION METACEUTIC APS (DK) 2021-12-02 WO claimed
EP-1067189-B1 GENE ENCODING FLAVONE SYNTHASE INTERNAT FLOWERS DEVELOPMENTS (AU) 2007-08-29 EP claimed
WO-2024095016-A1 COCOA-FREE CHOCOLATE NUKOKO LIMITED (GB) 2024-05-10 WO disclosed
WO-2024054415-A1 A COMBINATION OF SCYLLO-INOSITOL AND FLAVONES EIRGEN PHARMA, LTD. (US) 2024-03-14 WO disclosed
WO-2024054415-A1 A COMBINATION OF SCYLLO-INOSITOL AND FLAVONES EIRGEN PHARMA, LTD. (US) 2024-03-14 WO disclosed
WO-2024054791-A1 COMBINATION TREATMENT OF SCYLLO-INOSITOL AND VITAMIN D AND/OR OTHER VITAMINS OR ACTIVE INGREDIENTS TO TREAT COGNITIVE DISORDERS EIRGEN PHARMA, LTD. (IE) 2024-03-14 WO disclosed
EP-4156973-A1 NUTRACEUTICAL COMPOSITION METACEUTIC APS (DK) 2023-04-05 EP disclosed
US-20230073367-A1 Systems and Methods for Identifying Food Processing and Prescribing a Diet NORTHEASTERN UNIVERSITY 2023-03-09 US disclosed
US-20220411808-A1 NOVEL FLOWER COLOR AND COLOR INTENSITY ALLELE IN ANGELONIA ANGUSTIFOLIA BALL HORTICULTURAL COMPANY 2022-12-29 US disclosed
CN-110240582-B Flavone derivative with tumor cell inhibiting function and preparation method and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2022-11-01 CN disclosed
EP-1072265-A1 Use of plant polyphenols for treating iron overload MEDIS S.r.l. Medical Infusion Systems (IT) 2001-01-31 EP disclosed
WO-2001005981-A1 GENES CODING FOR FLAVONE SYNTHASES SUNTORY LIMITED (JP) 2001-01-25 WO disclosed
EP-1067189-A1 GENE ENCODING FLAVONE SYNTHASE SUNTORY LIMITED (JP) 2001-01-10 EP disclosed
WO-2000065073-A2 GENETIC SEQUENCE WHICH CODES FOR THE FLAVON SYNTHASE II ENZYME AND USE OF THE SAME MARTENS STEFAN (DE) 2000-11-02 WO disclosed
US-5023180-A Bradyrhizobium japonicum nodulation regulatory protein and gene LUBRIZOL GENETICS, INC. (US) 1991-06-11 US disclosed
EP-0269725-A4 BRADYRHIZOBIUM JAPONICUM NODULATION REGULATORY PROTEIN AND GENE. LUBRIZOL GENETICS INC (US) 1989-01-12 EP disclosed
US-4786498-A Process for the production of camomile extracts rich in flavones DEGUSSA AKTIENGESELLSCHAFT (DE) 1988-11-22 US disclosed
EP-0269725-A1 BRADYRHIZOBIUM JAPONICUM NODULATION REGULATORY PROTEIN AND GENE LUBRIZOL GENETICS INC. (US) 1988-06-08 EP disclosed
WO-1987007910-A1 BRADYRHIZOBIUM JAPONICUM NODULATION REGULATORY PROTEIN AND GENE LUBRIZOL GENETICS, INC. (US) 1987-12-30 WO disclosed