SCHEMBL3433244

SCHEMBL3433244

Cn1c(=O)c(C(F)(F)F)nc2cc(-c3cccc(OCC(F)(F)F)c3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.40
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
TGFBR1 P36897 2/20 0.39
CCKAR P32238 1/20 0.37
SLC5A1 P13866 3/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
TP53 P04637 1/20 0.37
NR3C1 P04150 1/20 0.36
ADORA2A P29274 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
BACE1 P56817 2/20 0.35
PPARG P37231 1/20 0.35
MAPT P10636 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3376646 0.87 MAPK14 (0.46) GRIN1GRIN2BTP53BACE1MAPK14
SCHEMBL3433242 0.85 MAPK14 (0.40) MAOAMAOBTGFBR1GRIN1GRIN2B
SCHEMBL3433378 0.82 TGFBR1 (0.51) TGFBR1GRIN1GRIN2BNR3C1MAPK14
SCHEMBL15147687 0.82 TGFBR1 (0.46) TGFBR1TP53NR3C1MAPTMAPK14
SCHEMBL3377364 0.78 SMN1; SMN2 (0.43) TP53
SCHEMBL3433560 0.78 MAPK14 (0.46) GRIN1GRIN2BTP53BACE1PPARG
SCHEMBL3474070 0.75 TGFBR1 (0.49) TGFBR1GRIN1GRIN2BNR3C1MAPK14
SCHEMBL3475344 0.74 KIT (0.48) GRIN1GRIN2BBACE1MAPK14
SCHEMBL20777094 0.71 FFAR4 (0.45) CTSAMAOBCCKARSLC5A1GRIN1
SCHEMBL3475092 0.71 ALDH1A1 (0.45) MAOAMAOBTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010053757-A1 2 -OXOQUINOXALIN BLOCKERS OF THE LATE SODIUM CHANNEL GILEAD PALO ALTO, INC. (US) 2010-05-14 WO claimed