SCHEMBL3433277

SCHEMBL3433277

C#Cc1ccc(Cl)cc1F

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
S1PR3 Q99500 7/20 0.34
TRPV4 Q9HBA0 1/20 0.33
TP53 P04637 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
VCAM1 P19320 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
S1PR1 P21453 4/20 0.32
S1PR2 O95136 1/20 0.32
S1PR4 O95977 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29932195 1.00 KMT2A (0.36) KMT2ACYP11B1CYP11B2PTGDR2S1PR3
SCHEMBL1544963 0.84 PTGDR2 (0.36) KMT2APTGDR2TP53CYP3A4TSHR
SCHEMBL6212336 0.77 PTGDR2 (0.38) KMT2ACYP11B1CYP11B2PTGDR2S1PR3
SCHEMBL496891 0.77 TRPV4 (0.57) CYP11B1CYP11B2S1PR3TRPV4VCAM1
SCHEMBL9996715 0.77 CYP11B1 (0.35) KMT2ACYP11B1CYP11B2PTGDR2S1PR3
SCHEMBL434666 0.76 ALDH1A1 (0.42) CYP11B1CYP11B2PTGDR2TRPV4TDP1
SCHEMBL30111761 0.76 ALDH1A1 (0.42) CYP11B1CYP11B2PTGDR2TRPV4TDP1
SCHEMBL2783347 0.76 TP53 (0.48) KMT2ATRPV4TP53CYP3A4TSHR
SCHEMBL19859678 0.76 ESR1 (0.42) CYP11B1CYP11B2
SCHEMBL16182687 0.74 HDAC8 (0.34) CYP11B1CYP11B2TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 86 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551834-B1 SUBSTITUTED QUINAZOLINONE COMPOUNDS NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-25 EP claimed
US-12528781-B2 Heterocyclic GLP-1 agonists GASHERBRUM BIO, INC. (US) 2026-01-20 US disclosed
EP-4638455-A1 HETEROCYCLIC GLP-1 AGONISTS Gasherbrum Bio, Inc. (US) 2025-10-29 EP disclosed
EP-4192831-B1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO INC (US) 2025-10-22 EP disclosed
US-20250145596-A1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO, INC. 2025-05-08 US disclosed
WO-2025034034-A1 NOVEL COMPOUND, AND PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF CANCER OR TUMORS COMPRISING SAME 주식회사 대웅제약 2025-02-13 WO disclosed
EP-4476213-A1 HETEROCYCLIC GLP-1 AGONISTS Gasherbrum Bio, Inc. (US) 2024-12-18 EP disclosed
CN-119072474-A Heterocyclic GLP-1 agonists 加舒布鲁姆生物公司 2024-12-03 CN disclosed
US-20240376061-A1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO, INC. 2024-11-14 US disclosed
US-12024507-B2 Compounds as GLP-1R agonists TERNS PHARMACEUTICALS, INC. (US) 2024-07-02 US disclosed
WO-2013186692-A1 TRIAZOLONE COMPOUNDS AS mPGES-1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2013-12-19 WO disclosed
WO-2013186692-A1 TRIAZOLONE COMPOUNDS AS mPGES-1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2013-12-19 WO disclosed
EP-1650284-B1 Liquid crystal composition containing an optical active compound and liquid crystal electro-optical element SEIMI CHEM KK (JP) 2008-04-30 EP disclosed
US-7108895-B2 Liquid crystal composition containing an optically active compound and liquid crystal electro-optical element SEIMI CHEMICAL CO., LTD. (JP) 2006-09-19 US disclosed
EP-1650284-A2 Liquid crystal composition containing an optical active compound and liquid crystal electro-optical element Seimi Chemical Co., Ltd. (JP) 2006-04-26 EP disclosed
EP-1650285-A2 Liquid crystal composition containing an optically active compound and liquid crystal electro-optical element Seimi Chemical Co., Ltd. (JP) 2006-04-26 EP disclosed
EP-1650286-A2 Liquid crystal composition containing an optically active compound and liquid crystal electro-optical element Seimi Chemical Co., Ltd. (JP) 2006-04-26 EP disclosed
US-20040079922-A1 Liquid crystal composition containing an optically active compound and liquid crystal electro-optical element SEIMI CHEMICAL CO., LTD. (JP) 2004-04-29 US disclosed
EP-1371712-A1 LIQUID-CRYSTAL COMPOSITION CONTAINING OPTICALLY ACTIVE COMPOUND AND LIQUID-CRYSTAL ELECTROOPTIC ELEMENT Seimi Chemical Co., Ltd. (JP) 2003-12-17 EP disclosed
WO-1997009881-A1 HERBICIDAL MIXTURES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1997-03-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12024507-B2 Compounds as GLP-1R agonists GLP1R, GIPR, GCGR KMT2A 4554/4885CYP11B1 1832/4885CYP11B2 2503/4885
US-12528781-B2 Heterocyclic GLP-1 agonists GLP1R, GIPR, VIP KMT2A 3022/4885CYP11B1 1495/4885CYP11B2 1987/4885
US-20250145596-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR KMT2A 3661/4885CYP11B1 917/4885CYP11B2 1402/4885
US-20240376061-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR KMT2A 4112/4885CYP11B1 1049/4885CYP11B2 1797/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.