SCHEMBL3434288

SCHEMBL3434288

CC(C)(C)OC(=O)NC(CC(=O)O)c1cc(-c2ccc([N+](=O)[O-])cc2)c(=O)[nH]n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
MAPT P10636 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
GAA P10253 2/20 0.38
DYRK1A Q13627 1/20 0.35
CYP1A2 P05177 1/20 0.35
GSK3B P49841 1/20 0.35
BCL2 P10415 1/20 0.34
BECN1 Q14457 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
TYMP P19971 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
AKR1C3 P42330 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL478795 0.93 MAPT (0.42) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL478796 0.93 MAPT (0.42) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL479148 0.89 F11 (0.44) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL479149 0.89 F11 (0.44) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL479109 0.85 PPARG (0.40) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL479110 0.85 PPARG (0.40) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL478745 0.84 F11 (0.46) MAPTGAAAAK1
SCHEMBL478746 0.84 F11 (0.46) MAPTGAAAAK1
SCHEMBL478943 0.83 ALDH1A1 (0.43) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL478941 0.83 ALDH1A1 (0.43) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2265601-A1 PYRIDAZINE DERIVATIVES AS FACTOR XIA INHIBITORS Bristol-Myers Squibb Company (US) 2010-12-29 EP disclosed
WO-2009114677-A1 PYRIDAZINE DERIVATIVES AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-09-17 WO disclosed