SCHEMBL3434951

SCHEMBL3434951

OC(c1ccccc1)c1cncnc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.67
CYP17A1 P05093 1/20 0.46
ATM Q13315 1/20 0.44
CFTR P13569 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
GOPC Q9HD26 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
GAA P10253 1/20 0.42
ALDH1A1 P00352 1/20 0.41
GRM5 P41594 1/20 0.40
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
LMNA P02545 3/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11138769 0.88 ATM (0.54) SMN1; SMN2CYP17A1ATMCYP11B1CYP11B2
SCHEMBL27306420 0.84 ATM (0.59) SMN1; SMN2CYP17A1ATMCYP11B1CYP11B2
SCHEMBL11134954 0.83 SMN1; SMN2 (0.49) SMN1; SMN2CYP17A1ATMLMNAHPGD
SCHEMBL28001042 0.80 SMN1; SMN2 (1.00) SMN1; SMN2CYP17A1CFTRSLC6A2SLC6A4
SCHEMBL30476558 0.80 SMN1; SMN2 (1.00) SMN1; SMN2CYP17A1CFTRSLC6A2SLC6A4
SCHEMBL30476552 0.80 SMN1; SMN2 (1.00) SMN1; SMN2CYP17A1CFTRSLC6A2SLC6A4
SCHEMBL477393 0.80 SMN1; SMN2 (1.00) SMN1; SMN2CYP17A1CFTRSLC6A2SLC6A4
SCHEMBL477633 0.80 SMN1; SMN2 (1.00) SMN1; SMN2CYP17A1CFTRSLC6A2SLC6A4
Diphenylmethanol SCHEMBL6434457 0.80 SMN1; SMN2 (0.61) SMN1; SMN2L3MBTL1LMNACA12CA1
Diphenylmethanol SCHEMBL41571 0.80 SMN1; SMN2 (0.61) SMN1; SMN2L3MBTL1LMNACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252296-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES Wyeth LLC (US) 2010-11-24 EP disclosed
WO-2009091788-A1 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-07-23 WO disclosed