SCHEMBL3435560

SCHEMBL3435560

Cc1c(C(=O)O)cccc1C(=O)N(C)Cc1ccc(F)c(-c2cccc(C=O)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TACR1 P25103 2/20 0.40
SCD5 Q86SK9 1/20 0.36
TRIM24 O15164 1/20 0.36
TRIM33 Q9UPN9 1/20 0.36
PPARG P37231 1/20 0.36
HPGD P15428 1/20 0.35
HSD17B1 P14061 2/20 0.34
HSD17B2 P37059 2/20 0.34
AOC3 Q16853 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PIN1 Q13526 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3433281 0.78 HPGD (0.50) KMT2AMEN1ALDH1A1TACR1HPGD
SCHEMBL1362397 0.78 ERN1 (0.47) KMT2AMEN1HSD17B1HSD17B2
SCHEMBL2559209 0.73 TRIM24 (0.53) ALDH1A1TRIM24TRIM33HPGD
SCHEMBL13761135 0.72 MAOA (0.40) ALDH1A1TRIM24TRIM33HPGD
SCHEMBL2560353 0.70 TRIM24 (0.63) KMT2AMEN1ALDH1A1TRIM24TRIM33
SCHEMBL6185510 0.68 AOC3 (0.45) KMT2AMEN1ALDH1A1AOC3
SCHEMBL4164586 0.67 KMT2A (0.66) KMT2AMEN1ALDH1A1HPGDHSP90AA1
SCHEMBL15332919 0.67 TRIM24 (0.62) TRIM24TRIM33
SCHEMBL2558013 0.67 TRIM24 (0.62) TRIM24TRIM33
SCHEMBL6715008 0.67 TRIM24 (0.57) ALDH1A1TRIM24TRIM33

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2249647-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS Glaxo Group Limited (GB) 2010-11-17 EP disclosed
WO-2009100168-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed