Valacyclovir

Valacyclovir

SCHEMBL34375

CC(C)[C@H](N)C(=O)OCCOCn1cnc2c(=O)nc(N)[nH]c21

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.72
MEN1 O00255 3/20 0.72
HBB P68871 2/20 0.71
MAPK1 P28482 1/20 0.71
PDE3A Q14432 1/20 0.50
PNP P00491 7/20 0.45
TSHR P16473 2/20 0.45
BLM P54132 2/20 0.45
USP2 O75604 1/20 0.45
EDNRA P25101 1/20 0.45
HTR2A P28223 1/20 0.45
RECQL P46063 1/20 0.45
HSD17B10 Q99714 1/20 0.45
HPRT1 P00492 4/20 0.41
POLG P54098 1/20 0.41
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
CYP3A4 P08684 1/20 0.37
NFKB1 P19838 1/20 0.37
VCP P55072 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Valacyclovir SCHEMBL4295083 1.00 KMT2A (0.72) KMT2AMEN1HBBMAPK1PDE3A
Valacyclovir SCHEMBL29689659 0.99 HBB (0.72) KMT2AMEN1HBBMAPK1PDE3A
Valacyclovir SCHEMBL1888797 0.98 KMT2A (0.69) KMT2AMEN1HBBMAPK1PDE3A
SCHEMBL23948433 0.86 KMT2A (0.53) KMT2AMEN1HBBMAPK1PDE3A
Valacyclovir SCHEMBL20570801 0.85 MEN1 (0.75) KMT2AMEN1HBBMAPK1PDE3A
Valganciclovir SCHEMBL336814 0.85 PDE3A (0.78) KMT2AMEN1HBBMAPK1PDE3A
Valacyclovir SCHEMBL4656778 0.84 MEN1 (1.00) KMT2AMEN1HBBMAPK1PDE3A
Valacyclovir SCHEMBL8444387 0.84 MEN1 (1.00) KMT2AMEN1HBBMAPK1PDE3A
Valacyclovir SCHEMBL13575743 0.84 MEN1 (1.00) KMT2AMEN1HBBMAPK1PDE3A
Valacyclovir SCHEMBL28644 0.84 MEN1 (1.00) KMT2AMEN1HBBMAPK1PDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 14378 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
EP-4094767-B1 NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO UNIV EMORY (US) 2026-05-20 EP claimed
US-20260124148-A1 POLYPEPTIDE FORMULATIONS FOR ORAL DELIVERY BHAMIS RES LABORATORY PVT LTD (IN) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4731194-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP Technologies, Inc. (US) 2026-04-29 EP claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-3790536-B1 NANOCONTAINERS FOR TRANSPORTING NONPOLAR, LIPOPHILIC SUBSTANCES SUCH AS ANTIBIOTICS KARLSRUHER INST TECHNOLOGIE (DE) 2026-04-22 EP claimed
US-20260102422-A1 4'-HALOGEN CONTAINING NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO UNIV EMORY (US) 2026-04-16 US claimed
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-12595280-B2 Phosphoramidates for the treatment of hepatitis B virus EMORY UNIVERSITY (US) 2026-04-07 US claimed
EP-0806943-A1 VALACICLOVIR TABLETS CONTAINING COLLOIDAL SILICON DIOXIDE THE WELLCOME FOUNDATION LIMITED (GB) 1997-11-19 EP claimed
EP-0804436-A1 GUANINE DERIVATIVE THE WELLCOME FOUNDATION LIMITED (GB) 1997-11-05 EP claimed
WO-1997026882-A1 NUCLEOSIDE ANALOGS IN COMBINATION THERAPY OF HERPES SIMPLEX INFECTIONS SMITHKLINE BEECHAM PLC (GB) 1997-07-31 WO claimed
WO-1997025989-A1 USE OF VALACICLOVIR FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF GENITAL HERPES BY A SINGLE DAILY APPLICATION GLAXO GROUP LIMITED (GB) 1997-07-24 WO claimed
WO-1996024354-A1 NOVEL PHARMACEUTICAL COMPOSITION ASTRA AKTIEBOLAG (SE) 1996-08-15 WO claimed
EP-0723448-A1 USE OF PENICLORIN FOR THE TREATMENT OF POSTTHERAPEUTIC NEURALGIA SMITHKLINE BEECHAM PLC (GB) 1996-07-31 EP claimed
WO-1996022291-A1 GUANINE DERIVATIVE THE WELLCOME FOUNDATION LIMITED (GB) 1996-07-25 WO claimed
WO-1996022082-A1 VALACICLOVIR TABLETS CONTAINING COLLOIDAL SILICON DIOXIDE THE WELLCOME FOUNDATION LIMITED (GB) 1996-07-25 WO claimed
WO-1995011027-A1 USE OF PENICLORIN FOR THE TREATMENT OF POSTTHERAPEUTIC NEURALGIA SMITHKLINE BEECHAM PLC (GB) 1995-04-27 WO claimed
WO-1995005179-A1 THERAPEUTIC COMBINATION CONTAINING AN ANTI-VARICELLA ZOSTER VIRUS COMPOUND AND LAMOTRIGINE THE WELLCOME FOUNDATION LIMITED (GB) 1995-02-23 WO claimed