SCHEMBL3444530

SCHEMBL3444530

CCn1nnc2c(Nc3cc(N)cc(Cl)c3)nc(NCC(C)N)nc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 10/20 0.44
CDK1 P06493 5/20 0.44
CCNB1 P14635 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 2/20 0.44
CCNB2 O95067 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CLK2 P49760 9/20 0.41
CLK4 Q9HAZ1 9/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3444882 0.91 CLK1 (0.46) CLK1CDK1CCNB1MEN1KMT2A
SCHEMBL3444409 0.88 CLK1 (0.48) CLK1CDK1CCNB1MEN1KMT2A
SCHEMBL3445942 0.87 CDK1 (0.52) CLK1CDK1CCNB1MEN1KMT2A
SCHEMBL3445810 0.87 CLK1 (0.47) CLK1CDK1CCNB1MEN1KMT2A
SCHEMBL3445484 0.87 KDM4E (0.49) CDK1MEN1KMT2AKDM4EALDH1A1
SCHEMBL3446013 0.85 BCDIN3D (0.41) CDK1MEN1KMT2AKDM4EALDH1A1
SCHEMBL3444649 0.85 CDK5 (0.40) CDK1MEN1KMT2AKDM4EALDH1A1
SCHEMBL3445162 0.83 MEN1 (0.50) MEN1KMT2AKDM4EALDH1A1TP53
SCHEMBL3444842 0.82 CDK1 (0.67) CLK1CDK1CCNB1MEN1KMT2A
SCHEMBL3444849 0.82 CDK1 (0.67) CLK1CDK1CCNB1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed