SCHEMBL3445458

SCHEMBL3445458

CCC(CO)Nc1nc(Nc2ccc(Cl)c(C(=O)O)c2)c2nn[nH]c2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 14/20 0.51
CDK5R1 Q15078 13/20 0.51
CDK1 P06493 6/20 0.51
KDM4E B2RXH2 3/20 0.43
MAPT P10636 2/20 0.43
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
CDK2 P24941 11/20 0.43
CCNA2 P20248 10/20 0.43
CCNA1 P78396 9/20 0.43
CCNE1 P24864 3/20 0.43
CCNB1 P14635 2/20 0.43
CCNB2 O95067 1/20 0.43
CCNE2 O96020 1/20 0.43
ALDH1A1 P00352 1/20 0.43
NTRK1 P04629 1/20 0.43
INSR P06213 1/20 0.43
PRKACA P17612 1/20 0.43
PRKACG P22612 1/20 0.43
PRKACB P22694 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446235 0.93 CDK5 (0.51) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3444046 0.90 CDK1 (0.50) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445184 0.87 CDK5 (0.66) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445461 0.86 CDK5 (0.46) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3444758 0.86 CDK5 (0.45) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3444318 0.84 CDK5 (0.45) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445866 0.83 CDK5 (0.47) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445114 0.82 CDK5 (0.62) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445554 0.81 CDK1 (0.46) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445923 0.81 KCNH3 (0.54) CDK5CDK5R1CDK1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed