SCHEMBL3445461

SCHEMBL3445461

CCC(CO)Nc1nc(Nc2ccc(Cl)c(C(=O)O)c2)c2[nH]nnc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 6/20 0.46
CDK5R1 Q15078 6/20 0.46
CDK1 P06493 5/20 0.46
KDM4E B2RXH2 4/20 0.39
MAPT P10636 3/20 0.39
NPC1 O15118 2/20 0.39
POLB P06746 2/20 0.39
CDK2 P24941 4/20 0.39
CCNA2 P20248 3/20 0.39
CCNA1 P78396 3/20 0.39
CCNE1 P24864 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CCNB2 O95067 1/20 0.39
CCNE2 O96020 1/20 0.39
NTRK1 P04629 1/20 0.39
INSR P06213 1/20 0.39
CCNB1 P14635 1/20 0.39
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446240 0.93 CDK5 (0.46) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3444051 0.90 CDK1 (0.46) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445187 0.88 CDK1 (0.61) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445458 0.86 CDK5 (0.51) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3444760 0.86 CDK5 (0.41) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3444324 0.84 CDK5 (0.41) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445871 0.84 CRHR1 (0.45) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445118 0.82 CDK5 (0.57) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445558 0.82 CDK1 (0.42) CDK5CDK5R1CDK1KDM4EMAPT
SCHEMBL3445927 0.82 KCNH3 (0.53) CDK5CDK5R1CDK1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed