SCHEMBL3446231

SCHEMBL3446231

C[Si](C)(C)C#Cc1cccc(CC(=O)O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 6/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
AKR1B1 P15121 1/20 0.46
NAPRT Q6XQN6 1/20 0.41
GAA P10253 3/20 0.41
TSHR P16473 2/20 0.41
NFKB1 P19838 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
ALDH1A1 P00352 1/20 0.41
PTGES O14684 2/20 0.40
KDM4E B2RXH2 1/20 0.40
RGS12 O14924 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
APEX1 P27695 1/20 0.40
THPO P40225 1/20 0.40
BLM P54132 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28027717 0.88 GRM5 (0.39) FFAR1CYP1A2CYP2C19NFKB1ALDH1A1
SCHEMBL5982854 0.85 ERCC1 (0.40) FFAR1PTGESLMNA
SCHEMBL4542339 0.83 FFAR1 (0.70) FFAR1CYP1A2CYP2C19AKR1B1PTGES
SCHEMBL3351697 0.81 FFAR1 (0.48) FFAR1TSHR
SCHEMBL21836127 0.81 PTGS1 (0.53) FFAR1AKR1B1GAATSHRNFKB1
SCHEMBL4945455 0.81 HDAC4 (0.39) FFAR1PTGESGABRA1GABRG2GABRB3
SCHEMBL8850812 0.80 HRH3 (0.47) PTGES
SCHEMBL27032998 0.80 NPC1 (0.43) FFAR1ALDH1A1PTGESHPGD
SCHEMBL1559856 0.80 FFAR1 (0.47) FFAR1
SCHEMBL3447198 0.80 FFAR1 (0.65) FFAR1AKR1B1GAATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010007482-A2 THIAZOLE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2010-01-21 WO disclosed