SCHEMBL4945455

SCHEMBL4945455

CON(C)C(=O)Cc1cccc(C#C[Si](C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
FFAR1 O14842 1/20 0.38
GRM5 P41594 2/20 0.36
ALOX5 P09917 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
PTGES O14684 5/20 0.35
LTB4R Q15722 3/20 0.35
LTB4R2 Q9NPC1 3/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRA6 Q16445 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4938489 0.85 FFAR1 (0.48) FFAR1PTGES
SCHEMBL1515861 0.81 MEP1A (0.46) FFAR1
SCHEMBL3446231 0.81 FFAR1 (0.49) FFAR1PTGESGABRA1GABRG2GABRB3
SCHEMBL4944372 0.80 PTGES (0.49) FFAR1GRM5SIGMAR1PTGES
SCHEMBL22607859 0.79 FFAR1 (0.38) FFAR1GRM5PTGES
SCHEMBL30267915 0.79 FFAR1 (0.38) FFAR1GRM5PTGES
SCHEMBL28027717 0.78 GRM5 (0.39) FFAR1GRM5PTGES
SCHEMBL1058423 0.76 CTBP2 (0.50) SIGMAR1LTB4RLTB4R2
SCHEMBL5982854 0.76 ERCC1 (0.40) FFAR1GRM5PTGES
SCHEMBL1515860 0.75 LMNA (0.43) HDAC4HDAC6ALOX5SIGMAR1LTB4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7465755-B2 Hydrazide derivatives as prostaglandin receptors modulators LABORATOIRES SERONO SA (CH) 2008-12-16 US disclosed
US-20070185191-A1 Hydrazide derivatives as prostaglandin receptors modulators APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (NL) 2007-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185191-A1 Hydrazide derivatives as prostaglandin receptors modulators PTGIR, HPGDS, PGF HDAC4 626/4885HDAC6 960/4885FFAR1 538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.