SCHEMBL3448383

SCHEMBL3448383

CC(=O)NCCNc1nc(Nc2ccc(F)c(Cl)c2)ncc1-c1cncc(C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
STK17A Q9UEE5 7/20 0.51
STK17B O94768 4/20 0.51
CSNK2A1 P68400 7/20 0.44
CSNK2A2 P19784 2/20 0.42
CSNK2B P67870 2/20 0.42
AURKA O14965 2/20 0.41
JAK2 O60674 2/20 0.41
AURKB Q96GD4 1/20 0.41
FLT1 P17948 1/20 0.41
JAK1 P23458 1/20 0.41
FLT4 P35916 1/20 0.41
BLK P51451 1/20 0.41
JAK3 P52333 1/20 0.41
TBK1 Q9UHD2 1/20 0.41
XDH P47989 1/20 0.41
SLC22A12 Q96S37 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3450308 0.91 STK17A (0.51) STK17ASTK17BCSNK2A1CSNK2A2CSNK2B
SCHEMBL3448722 0.90 STK17A (0.54) STK17ASTK17BJAK2FLT1JAK1
SCHEMBL3450274 0.90 STK17A (0.49) STK17ASTK17BCSNK2A1JAK2FLT1
SCHEMBL3450275 0.89 STK17A (0.47) STK17ASTK17BCSNK2A1AURKB
SCHEMBL3447250 0.88 CSNK2A1 (0.57) STK17ASTK17BCSNK2A1CSNK2A2CSNK2B
SCHEMBL3448505 0.88 CSNK2A1 (0.57) STK17ASTK17BCSNK2A1CSNK2A2CSNK2B
SCHEMBL3449309 0.87 STK17A (0.52) STK17ASTK17BCSNK2A1CSNK2A2CSNK2B
SCHEMBL3448962 0.87 STK17A (0.48) STK17ASTK17BCSNK2A1CSNK2A2CSNK2B
SCHEMBL3377446 0.87 CSNK2A1 (0.52) STK17ASTK17BCSNK2A1CSNK2A2CSNK2B
SCHEMBL3457207 0.87 CSNK2A1 (0.48) STK17ASTK17BCSNK2A1CSNK2A2CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF SDHA, SDHB, UROD STK17A 1984/4885STK17B 2457/4885CSNK2A1 1858/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.