SCHEMBL3450445

SCHEMBL3450445

FC(F)(F)c1cccc(Nc2nc(-c3ccccc3)cc(N3CCOCC3)n2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.65
SMG1 Q96Q15 2/20 0.65
USP2 O75604 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
IDH2 P48735 3/20 0.54
NPSR1 Q6W5P4 4/20 0.54
MAPT P10636 2/20 0.54
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
HSD17B10 Q99714 1/20 0.54
PIK3CA P42336 2/20 0.53
CNR2 P34972 1/20 0.53
RAF1 P04049 3/20 0.50
BRAF P15056 3/20 0.50
AIMP2 Q13155 1/20 0.49
AKT1 P31749 1/20 0.49
ATM Q13315 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
FLT1 P17948 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3451261 0.92 MTOR (0.63) MTORSMG1USP2SMN1; SMN2IDH2
SCHEMBL3451413 0.87 NPSR1 (0.67) SMG1NPSR1MAPTTSHRMAPK1
SCHEMBL18214299 0.86 MTOR (0.60) MTORSMG1USP2SMN1; SMN2IDH2
SCHEMBL3453662 0.86 IDH2 (0.67) MTORSMG1IDH2MAPT
SCHEMBL13127077 0.84 MAPT (0.64) MTORSMG1SMN1; SMN2NPSR1MAPT
SCHEMBL12485625 0.82 USP2 (0.60) MTORSMG1USP2SMN1; SMN2IDH2
SCHEMBL28449253 0.81 USP2 (0.78) USP2SMN1; SMN2IDH2MAPTPIK3CA
SCHEMBL3451414 0.81 PIK3CA (0.66) MTORSMG1USP2SMN1; SMN2IDH2
Hydrochloric Acid SCHEMBL17698146 0.81 USP2 (0.59) MTORSMG1USP2SMN1; SMN2IDH2
SCHEMBL3450413 0.80 ABL1 (0.56) MTORSMG1NPSR1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7820654-B2 Pyrimidine compounds, process for their preparation and compositions containing them DR. REDDY'S LABORATORIES LTD. (IN) 2010-10-26 US claimed
US-20060084645-A1 Novel pyrimidine compounds, process for their preparation and compositions containing them DR. REDDY'S LABORATORIES LTD. (IN) 2006-04-20 US claimed
US-7820654-B2 Pyrimidine compounds, process for their preparation and compositions containing them DR. REDDY'S LABORATORIES LTD. (IN) 2010-10-26 US disclosed
US-7820654-B2 Pyrimidine compounds, process for their preparation and compositions containing them DR. REDDY'S LABORATORIES LTD. (IN) 2010-10-26 US disclosed
US-7820654-B2 Pyrimidine compounds, process for their preparation and compositions containing them DR. REDDY'S LABORATORIES LTD. (IN) 2010-10-26 US disclosed
EP-1796673-A2 NOVEL PYRIMIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM Reddy US Therapeutics, Inc. (US) 2007-06-20 EP disclosed
US-20060084645-A1 Novel pyrimidine compounds, process for their preparation and compositions containing them DR. REDDY'S LABORATORIES LTD. (IN) 2006-04-20 US disclosed
WO-2006034473-A2 NOVEL PYRIMIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM REDDY US THERAPEUTICS, INC. (US) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060084645-A1 Novel pyrimidine compounds, process for their preparation and compositions containing them UMPS, DPYD, TYMS MTOR 1132/4885SMG1 947/4885USP2 3531/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.