SCHEMBL3451245

SCHEMBL3451245

COCCCNc1nc(Nc2ccc(F)c(Cl)c2)ncc1-c1cnc(OC)nc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
STK17A Q9UEE5 15/20 0.59
STK17B O94768 9/20 0.59
BCL6 P41182 4/20 0.47
JAK2 O60674 1/20 0.43
FLT1 P17948 1/20 0.43
JAK1 P23458 1/20 0.43
FLT4 P35916 1/20 0.43
BLK P51451 1/20 0.43
JAK3 P52333 1/20 0.43
TBK1 Q9UHD2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13310862 0.90 STK17A (0.57) STK17ASTK17BBCL6
SCHEMBL13310753 0.89 STK17A (0.57) STK17ASTK17BBCL6
SCHEMBL13420401 0.85 STK17A (0.52) STK17ASTK17BBCL6
SCHEMBL13310837 0.84 STK17A (0.54) STK17ASTK17BBCL6
SCHEMBL13311472 0.84 STK17A (0.50) STK17ASTK17BBCL6JAK3
SCHEMBL13311405 0.83 STK17A (0.48) STK17ASTK17BBCL6
SCHEMBL3450356 0.83 STK17A (0.48) STK17ASTK17BBCL6JAK3
SCHEMBL3450877 0.83 STK17A (0.52) STK17ASTK17BBCL6JAK2FLT1
SCHEMBL13312760 0.83 STK17A (0.52) STK17ASTK17BBCL6JAK2FLT1
SCHEMBL3449939 0.83 STK17A (0.52) STK17ASTK17BBCL6JAK2FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF SDHA, SDHB, UROD STK17A 1984/4885STK17B 2457/4885BCL6 3290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.