SCHEMBL3455376

SCHEMBL3455376

COC(=O)CC1Nc2ccccc2CN(C)C1=O

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 16/20 0.49
ITGAV P06756 13/20 0.49
ITGA2B P08514 10/20 0.47
BRD4 O60885 1/20 0.44
CREBBP Q92793 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8526495 1.00 ITGB3 (0.49) ITGB3ITGAVITGA2BBRD4CREBBP
SCHEMBL8503077 0.86 ITGB3 (0.61) ITGB3ITGAVITGA2B
SCHEMBL8187415 0.84 ITGB3 (0.49) ITGB3ITGAVITGA2B
SCHEMBL8525346 0.83 ITGB3 (0.48) ITGB3ITGAVITGA2B
SCHEMBL7909994 0.83 BRD4 (0.49) ITGB3ITGAVITGA2BBRD4
SCHEMBL7919360 0.83 ITGB3 (0.48) ITGB3ITGAVITGA2B
SCHEMBL4024909 0.82 ITGB3 (0.57) ITGB3ITGAVITGA2B
SCHEMBL4023860 0.82 ITGB3 (0.57) ITGB3ITGAVITGA2B
SCHEMBL5155928 0.82 ITGB3 (0.57) ITGB3ITGAVITGA2B
SCHEMBL7366349 0.81 ITGB3 (0.58) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2196458-A1 Process for obtaining enantiomerically enriched pyrazole derivatives Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-06-16 EP disclosed
US-6225465-B1 REACTING BENZOAZEPINE OR BENZODIAZEPINE DERIVATIVE WITH PROTECTED AMINE IN PRESENCE OF PALLADIUM CATALYST IN PRESENCE OF CARBON MONOXIDE, REMOVING PROTECTING GROUPS SMITHKLINE BEECHAM PLC (GB) 2001-05-01 US disclosed
WO-2000063186-A1 PROCESS AND INTERMEDIATES FOR PREPARING BENZODIAZEPINES SMITHKLINE BEECHAM PLC (GB) 2000-10-26 WO disclosed
EP-1019383-A2 PROCESS FOR THE AMINOCARBONYLATION OF BENZAZEPINES AND BENZODIAZEPINES SMITHKLINE BEECHAM PLC (GB) 2000-07-19 EP disclosed
EP-0964928-A1 ENZYMATIC RESOLUTION OF BENZODIAZEPINE-ACETIC ACID ESTERS WITH A LIPASE SMITHKLINE BEECHAM PLC (GB) 1999-12-22 EP disclosed
WO-1998029561-A1 ENZYMATIC RESOLUTION OF BENZODIAZEPINE-ACETIC ACID ESTERS WITH A LIPASE SMITHKLINE BEECHAM PLC (GB) 1998-07-09 WO disclosed
WO-1997024336-A2 PROCESS FOR THE AMINOCARBONYLATION OF BENZAZEPINES AND BENZODIAZEPINES SMITHKLINE BEECHAM PLC (GB) 1997-07-10 WO disclosed