SCHEMBL3456743

SCHEMBL3456743

CC(C)Cc1ccc(C(=O)NN)cc1.C[SiH](C)OC(c1ccc(C(=O)O)cc1)C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 3/20 0.41
CXCR2 P25025 3/20 0.41
PTGS1 P23219 4/20 0.40
PTGS2 P35354 4/20 0.40
LMNA P02545 2/20 0.40
CYP2C9 P11712 2/20 0.40
AKR1C3 P42330 2/20 0.40
NR1H4 Q96RI1 2/20 0.40
ALB P02768 1/20 0.40
ESR1 P03372 1/20 0.40
ALOX5 P09917 1/20 0.40
RARB P10826 1/20 0.40
ADRB3 P13945 1/20 0.40
NFKB1 P19838 1/20 0.40
HTR2A P28223 1/20 0.40
NR1I3 Q14994 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40
CXCL8 P10145 1/20 0.40
TSHR P16473 1/20 0.40
AKR1C2 P52895 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809114 0.87 MAPT (0.46) LMNANR1H4BLMPMP22
SCHEMBL6671659 0.80 NR1H4 (0.42) NR1H4RARBTSHREPHX2SMN1; SMN2
SCHEMBL3456546 0.76 BLM (0.53) CXCR1CXCR2PTGS1PTGS2LMNA
SCHEMBL3456745 0.74 NR1H4 (0.41) CXCR1CXCR2PTGS1PTGS2LMNA
SCHEMBL17111856 0.73 RXRA (0.41) PTGS1LMNAAKR1C3NR1H4TSHR
SCHEMBL27959311 0.71 PTGS1 (0.60) CXCR1CXCR2PTGS1PTGS2LMNA
SCHEMBL452233 0.71 PTGS1 (0.60) CXCR1CXCR2PTGS1PTGS2LMNA
SCHEMBL5973107 0.71 CA1 (0.44) CYP2C9TSHRGAA
SCHEMBL977243 0.71 PPARA (0.52)
SCHEMBL8793404 0.70 PTGS1 (0.61) CXCR1CXCR2PTGS1PTGS2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258700-A1 Cycloalkylamino acid derivatives and pharmaceutical compositions thereof Pfizer Products Inc. (US) 2010-12-08 EP disclosed