SCHEMBL3456745

SCHEMBL3456745

CC(C)(C)[SiH2]OC(C)(C)c1ccc(C(=O)O)cc1.CC(C)Cc1ccc(C(=O)NN)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.41
EPHX2 P34913 1/20 0.41
ALDH1A1 P00352 4/20 0.39
NR4A2 P43354 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
MAPT P10636 5/20 0.37
ANPEP P15144 1/20 0.36
ENPEP Q07075 1/20 0.36
CXCR1 P25024 1/20 0.36
CXCR2 P25025 1/20 0.36
ACACB O00763 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
LMNA P02545 1/20 0.35
ALB P02768 1/20 0.35
ESR1 P03372 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3456546 0.77 BLM (0.53) ALDH1A1MAPTCXCR1CXCR2CA1
SCHEMBL3456743 0.74 CXCR1 (0.41) NR1H4EPHX2RXRARXRBCXCR1
SCHEMBL5438501 0.73 CA1 (0.44) ALDH1A1MAPTCA1CA2MAPK1
SCHEMBL27959311 0.72 PTGS1 (0.60) ALDH1A1ANPEPENPEPCXCR1CXCR2
SCHEMBL452233 0.72 PTGS1 (0.60) ALDH1A1ANPEPENPEPCXCR1CXCR2
SCHEMBL978696 0.71 ESR1 (0.37) NR1H4ALDH1A1MAPTACACBLMNA
SCHEMBL10749840 0.71 NR1H4 (0.46) NR1H4EPHX2ALDH1A1NR4A2RXRA
SCHEMBL977245 0.70 PPARA (0.53)
SCHEMBL9369118 0.68 ADRB3 (0.56) ALDH1A1RXRARXRBMAPTANPEP
SCHEMBL72425 0.67 MPO (0.67) ALDH1A1MAPTCA1CA2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258700-A1 Cycloalkylamino acid derivatives and pharmaceutical compositions thereof Pfizer Products Inc. (US) 2010-12-08 EP disclosed