SCHEMBL3456772

SCHEMBL3456772

Cc1cc(C(F)(F)F)nn1-c1nc(Nc2ccc(F)c(Cl)c2)ncc1-c1cc(C(=O)O)c(=O)n(C)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SYK P43405 8/20 0.38
EGFR P00533 3/20 0.36
PDGFRB P09619 1/20 0.36
FGFR1 P11362 1/20 0.36
SRC P12931 1/20 0.36
PDGFRA P16234 1/20 0.36
STAT5A P42229 1/20 0.36
ACVR1 Q04771 1/20 0.36
PKMYT1 Q99640 1/20 0.36
AXL P30530 2/20 0.35
MAPK14 Q16539 1/20 0.35
KCNN3 Q9UGI6 1/20 0.35
XDH P47989 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
STK17A Q9UEE5 1/20 0.34
ULK1 O75385 1/20 0.34
WEE1 P30291 1/20 0.34
TYRO3 Q06418 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3447261 0.93 EGFR (0.36) SYKEGFRPDGFRBFGFR1SRC
SCHEMBL3448714 0.91 SYK (0.38) SYKEGFRPDGFRBFGFR1SRC
SCHEMBL3448963 0.91 SYK (0.36) SYKEGFRPDGFRBFGFR1SRC
SCHEMBL3448666 0.90 SCN9A (0.39)
SCHEMBL3449131 0.89 SYK (0.37) SYKEGFRAXL
SCHEMBL3447298 0.88 RAF1 (0.38) SYKEGFRPDGFRBFGFR1SRC
SCHEMBL3450229 0.87 SYK (0.39) SYKEGFRPDGFRBFGFR1SRC
SCHEMBL3452706 0.87 SYK (0.42) SYK
SCHEMBL3454800 0.87 SYK (0.42) SYKEGFRAXLWEE1
SCHEMBL3448336 0.87 SYK (0.38) SYKEGFRKCNN3XDHSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF SDHA, SDHB, UROD SYK 804/4885EGFR 2771/4885PDGFRB 2785/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.