SCHEMBL3463240

SCHEMBL3463240

COCC(C)Oc1cc(Oc2cnc(C(=O)N3CCN(C)CC3)cn2)cc(-c2ccc(C(=O)OCc3ccccc3)[nH]2)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GCK P35557 16/20 0.47
KCNH2 Q12809 5/20 0.38
CYP1A2 P05177 1/20 0.35
ABCB1 P08183 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35
HPGDS O60760 1/20 0.34
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
NPC1 O15118 1/20 0.33
SCN7A Q01118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1055145 1.00 GCK (0.47) GCKKCNH2CYP1A2ABCB1CYP3A4
SCHEMBL1056454 0.84 GCK (0.52) GCKKCNH2CYP1A2ABCB1CYP3A4
SCHEMBL421885 0.82 GCK (0.43) GCKKCNH2RARARARB
SCHEMBL2669700 0.81 GCK (0.52) GCKKCNH2CYP1A2ABCB1CYP3A4
SCHEMBL423126 0.81 GCK (0.52) GCKKCNH2CYP1A2ABCB1CYP3A4
SCHEMBL13127258 0.80 GCK (0.57) GCKKCNH2CYP1A2ABCB1CYP3A4
SCHEMBL425598 0.80 GCK (0.41) GCKKCNH2RARARARB
SCHEMBL428556 0.79 GCK (0.48) GCKKCNH2CYP1A2ABCB1CYP3A4
SCHEMBL423252 0.77 GCK (0.41) GCKKCNH2
SCHEMBL426478 0.77 MMP2 (0.41) GCKCYP3A4RARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239253-A1 NOVEL PHENYLPYRROLE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-10-13 EP disclosed