SCHEMBL3463404

SCHEMBL3463404

CCc1ncc(-c2cnc(Nc3ccc(F)c(Cl)c3)nc2NC2CCOC2)cc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TYRO3 Q06418 7/20 0.42
SYK P43405 4/20 0.42
STK17A Q9UEE5 2/20 0.42
STK17B O94768 1/20 0.42
SELP P16109 1/20 0.41
CSNK2A1 P68400 1/20 0.40
LRRK2 Q5S007 1/20 0.40
EGFR P00533 3/20 0.40
AXL P30530 5/20 0.40
MERTK Q12866 4/20 0.40
BRAF P15056 1/20 0.40
ITK Q08881 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3463408 1.00 TYRO3 (0.42) TYRO3SYKSTK17ASTK17BSELP
SCHEMBL3448900 0.84 CSNK2A1 (0.46) TYRO3SYKSELPCSNK2A1LRRK2
SCHEMBL3449243 0.84 CSNK2A1 (0.46) TYRO3SYKSELPCSNK2A1LRRK2
SCHEMBL3451208 0.81 EGFR (0.44) TYRO3STK17ASTK17BLRRK2EGFR
SCHEMBL3447987 0.81 EGFR (0.44) TYRO3STK17ASTK17BLRRK2EGFR
SCHEMBL3463402 0.81 TYRO3 (0.43) TYRO3SYKSTK17ASELPLRRK2
SCHEMBL3450787 0.81 EGFR (0.41) TYRO3SYKSTK17ASELPLRRK2
SCHEMBL3450789 0.81 EGFR (0.41) TYRO3SYKSTK17ASELPLRRK2
SCHEMBL3450057 0.80 IRAK4 (0.42) TYRO3SYKSELPCSNK2A1LRRK2
SCHEMBL3449272 0.79 EGFR (0.43) TYRO3SYKSELPCSNK2A1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB 2010-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137313-A1 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF SDHA, SDHB, UROD TYRO3 2798/4885SYK 804/4885STK17A 1984/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.