SCHEMBL3467478

SCHEMBL3467478

COc1ccc(NC(=O)c2cn(CCCC(=O)NO)c3ccc(OC)cc3c2=O)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.54
HDAC3 O15379 4/20 0.54
HDAC6 Q9UBN7 4/20 0.54
GAA P10253 2/20 0.54
TP53 P04637 3/20 0.53
TDP1 Q9NUW8 3/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HDAC1 Q13547 3/20 0.51
HDAC2 Q92769 3/20 0.51
HDAC8 Q9BY41 3/20 0.51
HDAC4 P56524 2/20 0.51
HDAC7 Q8WUI4 2/20 0.51
HDAC10 Q969S8 2/20 0.51
HDAC11 Q96DB2 2/20 0.51
HDAC9 Q9UKV0 2/20 0.51
HDAC5 Q9UQL6 2/20 0.51
KMT2A Q03164 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7912521 0.96 HDAC3 (0.59) MAPTHDAC3HDAC6GAATP53
SCHEMBL3467483 0.91 GAA (0.60) MAPTHDAC3HDAC6GAATP53
SCHEMBL3468407 0.91 MAPT (0.56) MAPTHDAC3HDAC6GAATP53
SCHEMBL3467874 0.91 HDAC6 (0.57) MAPTHDAC3HDAC6GAATP53
SCHEMBL3467664 0.90 HDAC6 (0.54) MAPTHDAC3HDAC6GAATP53
SCHEMBL3467891 0.90 HDAC6 (0.54) MAPTHDAC3HDAC6GAATP53
SCHEMBL3467448 0.89 GAA (0.54) MAPTHDAC3HDAC6GAATP53
SCHEMBL3468139 0.87 CNR2 (0.58) HDAC3HDAC6HDAC1HDAC2HDAC8
SCHEMBL3467591 0.87 HDAC3 (0.51) MAPTHDAC3HDAC6GAASMN1; SMN2
SCHEMBL7921598 0.87 HDAC6 (0.55) HDAC3HDAC6GAATP53TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO claimed
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed