SCHEMBL3467591

SCHEMBL3467591

COc1ccc2c(c1)c(=O)c(C(=O)Nc1ccc(N3CCCCC3)cc1)cn2CCCCCC(=O)NO

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.51
HDAC6 Q9UBN7 3/20 0.51
MAPT P10636 8/20 0.48
CNR1 P21554 3/20 0.46
CNR2 P34972 3/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
GAA P10253 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
ALDH1A1 P00352 3/20 0.45
RAB9A P51151 3/20 0.45
KMT2A Q03164 2/20 0.45
NR4A1 P22736 1/20 0.45
MCL1 Q07820 1/20 0.45
LMNA P02545 2/20 0.44
NPC1 O15118 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
QSOX1 O00391 1/20 0.44
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7912521 0.90 HDAC3 (0.59) HDAC3HDAC6MAPTCNR1CNR2
SCHEMBL3468407 0.87 MAPT (0.56) HDAC3HDAC6MAPTHDAC1HDAC2
SCHEMBL3467483 0.87 GAA (0.60) HDAC3HDAC6MAPTCNR1CNR2
SCHEMBL3467874 0.87 HDAC6 (0.57) HDAC3HDAC6MAPTCNR1CNR2
SCHEMBL3467478 0.87 MAPT (0.54) HDAC3HDAC6MAPTCNR1CNR2
SCHEMBL3467891 0.85 HDAC6 (0.54) HDAC3HDAC6MAPTCNR1CNR2
SCHEMBL3467664 0.85 HDAC6 (0.54) HDAC3HDAC6MAPTCNR1CNR2
SCHEMBL3467448 0.84 GAA (0.54) HDAC3HDAC6MAPTCNR1CNR2
SCHEMBL7921598 0.83 HDAC6 (0.55) HDAC3HDAC6CNR1CNR2HDAC1
SCHEMBL3467570 0.82 HDAC6 (0.54) HDAC3HDAC6MAPTCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed