SCHEMBL3467448

SCHEMBL3467448

COc1ccc(NC(=O)c2cn(CCCCCC(=O)NO)c3ccc(F)cc3c2=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.54
HDAC3 O15379 5/20 0.51
HDAC6 Q9UBN7 5/20 0.51
MAPT P10636 5/20 0.51
HDAC1 Q13547 5/20 0.50
HDAC2 Q92769 5/20 0.50
HDAC8 Q9BY41 4/20 0.50
HDAC4 P56524 3/20 0.50
HDAC7 Q8WUI4 3/20 0.50
HDAC10 Q969S8 3/20 0.50
HDAC11 Q96DB2 3/20 0.50
HDAC9 Q9UKV0 3/20 0.50
HDAC5 Q9UQL6 3/20 0.50
KMT2A Q03164 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
POLB P06746 2/20 0.49
TUBB4A P04350 1/20 0.49
TUBB P07437 1/20 0.49
TUBA3C P0DPH7 1/20 0.49
TUBA1B P68363 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467483 0.95 GAA (0.60) GAAHDAC3HDAC6MAPTHDAC1
SCHEMBL7912521 0.93 HDAC3 (0.59) GAAHDAC3HDAC6MAPTHDAC1
SCHEMBL3467960 0.92 HDAC1 (0.51) GAAHDAC3HDAC6MAPTHDAC1
SCHEMBL3467478 0.89 MAPT (0.54) GAAHDAC3HDAC6MAPTHDAC1
SCHEMBL3467582 0.89 HDAC1 (0.55) GAAHDAC3HDAC6MAPTHDAC1
SCHEMBL3476785 0.88 TP53 (0.51) GAAHDAC3HDAC6MAPTHDAC1
SCHEMBL3467644 0.88 HDAC1 (0.52) HDAC3HDAC6HDAC1HDAC2HDAC8
SCHEMBL3468407 0.88 MAPT (0.56) GAAHDAC3HDAC6MAPTHDAC1
SCHEMBL3467092 0.88 CNR2 (0.46) HDAC3HDAC6MAPTHDAC1HDAC2
SCHEMBL3467874 0.88 HDAC6 (0.57) GAAHDAC3HDAC6MAPTHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO claimed
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed