SCHEMBL3467644

SCHEMBL3467644

O=C(CCCCCn1cc(C(=O)Nc2ccccc2)c(=O)c2cc(F)ccc21)NO

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 15/20 0.52
HDAC6 Q9UBN7 14/20 0.52
HDAC3 O15379 4/20 0.48
HDAC4 P56524 4/20 0.48
HDAC7 Q8WUI4 4/20 0.48
HDAC11 Q96DB2 4/20 0.48
HDAC8 Q9BY41 4/20 0.48
HDAC9 Q9UKV0 4/20 0.48
HDAC5 Q9UQL6 4/20 0.48
HDAC2 Q92769 4/20 0.48
EGFR P00533 3/20 0.48
HDAC10 Q969S8 3/20 0.48
CNR2 P34972 2/20 0.47
CNR1 P21554 1/20 0.47
KDM4E B2RXH2 1/20 0.46
BRD4 O60885 1/20 0.46
NCOR1 O75376 1/20 0.46
NR1I2 O75469 1/20 0.46
CYP3A4 P08684 1/20 0.46
LTA4H P09960 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467960 0.94 HDAC1 (0.51) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL7919685 0.91 HDAC1 (0.47) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3467582 0.91 HDAC1 (0.55) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3467463 0.89 CNR2 (0.58) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3467448 0.88 GAA (0.54) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3467092 0.88 CNR2 (0.46) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3467928 0.88 HDAC1 (0.60) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3467867 0.87 MAPT (0.50) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3467874 0.86 HDAC6 (0.57) HDAC1HDAC6HDAC3HDAC8HDAC2
SCHEMBL3467483 0.85 GAA (0.60) HDAC1HDAC6HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO claimed
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed